SCHEMBL7584411

SCHEMBL7584411

C=C1[C@@H](c2ccc(OC)cc2)[C@@](C)(c2cccc(C#N)c2)NC(=N)N1C

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32
BACE1 P56817 1/20 0.32
SNCA P37840 1/20 0.31
MCHR1 Q99705 2/20 0.31
NPBWR1 P48145 1/20 0.31
USP2 O75604 4/20 0.31
ALDH1A1 P00352 3/20 0.31
TSHR P16473 3/20 0.31
CYP3A4 P08684 3/20 0.31
CYP1A2 P05177 2/20 0.31
MAPK1 P28482 1/20 0.31
GRIN1 Q05586 1/20 0.30
GRIN2B Q13224 1/20 0.30
KDM4E B2RXH2 1/20 0.30
LMNA P02545 1/20 0.30
GAA P10253 1/20 0.30
HTT P42858 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7582435 0.91 BACE1 (0.34) BACE1ALDH1A1
SCHEMBL7589796 0.90 ALDH1A1 (0.32) KMT2AMEN1MAPTBACE1ALDH1A1
SCHEMBL7589838 0.89 BACE1 (0.36) BACE1CYP3A4
SCHEMBL7541955 0.88 BACE1 (0.36) KMT2AMEN1MAPTBACE1MCHR1
SCHEMBL13054897 0.88 BACE1 (0.36) KMT2AMEN1MAPTBACE1MCHR1
SCHEMBL7584854 0.87 BACE1 (0.30) BACE1
SCHEMBL7582630 0.86 KDM1A (0.31) BACE1SLC6A2SLC6A4
SCHEMBL7584371 0.85 BACE1 (0.31) BACE1
SCHEMBL7584231 0.85 ELANE (0.33) BACE1CYP3A4KDM4EHTT
SCHEMBL7581043 0.85 BACE1 (0.31) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8183252-B2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2012-05-22 US disclosed