SCHEMBL7584472

SCHEMBL7584472

O=C(O)CC(c1ccc(-c2ccccc2)c(F)c1)N1CCN(CCCC2=CC=C3CCCNC3N2)C1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 10/20 0.47
ITGB3 P05106 8/20 0.47
ITGB8 P26012 6/20 0.44
ITGB6 P18564 5/20 0.44
ITGA5 P08648 4/20 0.39
ITGB1 P05556 1/20 0.39
ITGA2B P08514 1/20 0.39
FFAR1 O14842 1/20 0.35
PTGS1 P23219 3/20 0.31
MEN1 O00255 2/20 0.31
PTGS2 P35354 2/20 0.31
KMT2A Q03164 2/20 0.31
FABP2 P12104 1/20 0.31
TSHR P16473 1/20 0.31
AKR1C4 P17516 1/20 0.31
ADRA2B P18089 1/20 0.31
CHRM3 P20309 1/20 0.31
HTR2C P28335 1/20 0.31
DRD3 P35462 1/20 0.31
AKR1C3 P42330 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7596086 1.00 ITGAV (0.47) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7597852 1.00 ITGAV (0.47) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7559347 0.88 ITGAV (0.49) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7597015 0.87 ITGAV (0.54) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7577451 0.87 ITGAV (0.54) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7601055 0.87 ITGAV (0.54) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL4367915 0.86 ITGAV (0.44) ITGAVITGB3ITGB8ITGB6FFAR1
SCHEMBL7592559 0.83 ITGAV (0.63) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7553084 0.83 ITGAV (0.63) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7595642 0.83 ITGAV (0.63) ITGAVITGB3ITGB8ITGB6ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040111-A1 INTEGRIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2000-10-04 EP claimed
WO-1999031099-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO claimed
EP-1040111-A1 INTEGRIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2000-10-04 EP disclosed
WO-1999031099-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO disclosed