SCHEMBL7585475

SCHEMBL7585475

O=CCCc1cc(F)c(OCCCN2CCN(c3cccc4ccsc34)CC2)c(F)c1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.51
HTR2A P28223 7/20 0.51
HTR1A P08908 6/20 0.51
KCNH2 Q12809 5/20 0.39
SLC6A4 P31645 2/20 0.39
HRH1 P35367 3/20 0.38
HRH3 Q9Y5N1 3/20 0.38
ADRA1A P35348 2/20 0.38
ADRA1B P35368 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7128893 0.84 HTR2A (0.55) DRD2HTR2AHTR1AKCNH2SLC6A4
SCHEMBL7127886 0.81 HTR1A (0.52) DRD2HTR2AHTR1AKCNH2SLC6A4
SCHEMBL7119229 0.80 HTR2A (0.58) DRD2HTR2AHTR1AKCNH2SLC6A4
SCHEMBL7119324 0.80 HTR2A (0.52) DRD2HTR2AHTR1AKCNH2SLC6A4
SCHEMBL7117583 0.78 DRD2 (0.55) DRD2HTR2AHTR1AKCNH2SLC6A4
SCHEMBL7118961 0.78 HTR2A (0.55) DRD2HTR2AHTR1AKCNH2SLC6A4
SCHEMBL7124105 0.78 HTR1A (0.55) DRD2HTR2AHTR1AKCNH2SLC6A4
SCHEMBL7123026 0.76 DRD2 (0.55) DRD2HTR2AHTR1AKCNH2SLC6A4
SCHEMBL7121850 0.76 HTR2A (0.56) DRD2HTR2AHTR1ASLC6A4
SCHEMBL7120429 0.76 DRD2 (0.52) DRD2HTR2AHTR1AKCNH2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1246820-A1 NOVEL HETEROARYL DERIVATIVES, THEIR PREPARATION AND USE H. LUNDBECK A/S (DK) 2002-10-09 EP disclosed
WO-2001049683-A1 NOVEL HETEROARYL DERIVATIVES, THEIR PREPARATION AND USE H. LUNDBECK A/S (DK) 2001-07-12 WO disclosed