SCHEMBL7586110

SCHEMBL7586110

CN(CCc1ccccc1)CC1=C(c2cccc(O)c2)c2ccccc2CCC1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 15/20 0.41
OPRM1 P35372 14/20 0.41
OPRD1 P41143 12/20 0.41
DRD2 P14416 5/20 0.41
DRD3 P35462 5/20 0.41
ESR1 P03372 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8018024 0.99 OPRK1 (0.43) OPRK1OPRM1OPRD1DRD2DRD3
SCHEMBL7588566 0.90 G6PC1 (0.41) OPRK1OPRM1OPRD1ESR1
Hydrochloric Acid SCHEMBL8017509 0.89 G6PC1 (0.41) OPRK1OPRM1OPRD1ESR1
SCHEMBL7584182 0.85 ESR1 (0.40) OPRK1OPRD1ESR1
SCHEMBL7591956 0.85 CYP2D6 (0.45)
Hydrochloric Acid SCHEMBL8011601 0.84 ESR1 (0.39) OPRK1OPRD1ESR1
Hydrochloric Acid SCHEMBL8014130 0.84 CYP2D6 (0.44)
SCHEMBL7587127 0.83 CHRNB4 (0.40) OPRK1OPRD1DRD2ESR1
SCHEMBL7587120 0.83 CHRNB4 (0.40) OPRK1OPRD1DRD2ESR1
SCHEMBL7606326 0.82 BCHE (0.42) OPRK1OPRM1OPRD1DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0864559-B1 Substituted amino compounds and their use as analgesic active substances GRUENENTHAL GMBH (DE) 2002-06-05 EP disclosed
EP-0864559-A1 Substituted amino compounds and their use as analgesic active substances Grünenthal GmbH (DE) 1998-09-16 EP disclosed