SCHEMBL758648

SCHEMBL758648

CN(c1cc[c]cc1)c1nc2ccccc2[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C19 P33261 1/20 0.50
BCHE P06276 1/20 0.49
ACHE P22303 1/20 0.49
ALDH1A1 P00352 4/20 0.43
HPGD P15428 1/20 0.43
MCL1 Q07820 1/20 0.43
POLB P06746 1/20 0.42
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
PKM P14618 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ABCB11 O95342 1/20 0.42
TP53 P04637 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HSD17B10 Q99714 1/20 0.42
DDAH1 O94760 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11303623 0.87 LMNA (0.56) LMNACYP1A2CYP2D6CYP2C19BCHE
SCHEMBL29025770 0.81 LMNA (0.61) LMNACYP1A2CYP2D6CYP2C19BCHE
SCHEMBL11100536 0.81 LMNA (0.50) LMNACYP1A2CYP2D6CYP2C19BCHE
SCHEMBL1268888 0.79 F2 (0.52) LMNACYP1A2CYP2D6CYP2C19BCHE
SCHEMBL358399 0.76 LMNA (0.62) LMNACYP1A2CYP2D6CYP2C19BCHE
SCHEMBL5562226 0.76 CHEK2 (0.54) LMNACYP1A2CYP2D6CYP2C19BCHE
SCHEMBL2001474 0.75 LMNA (0.47) LMNACYP1A2CYP2D6CYP2C19BCHE
Hydrochloric Acid SCHEMBL270477 0.74 LMNA (0.66) LMNACYP1A2CYP2D6CYP2C19BCHE
Hydrochloric Acid SCHEMBL270476 0.74 LMNA (0.66) LMNACYP1A2CYP2D6CYP2C19BCHE
Hydrochloric Acid SCHEMBL20291494 0.74 LMNA (0.66) LMNACYP1A2CYP2D6CYP2C19BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101346355-B Improved process for preparing salts of 4- (benzimidazolylmethylamino) -benzamidines BOEHRINGER INGELHEIM INT 2012-09-05 CN disclosed
CN-1972919-B Method for producing 4-(benzimidazolylmethylamino)-benzamidines BOEHRINGER INGELHEIM INT 2012-06-27 CN disclosed
EP-1847534-B9 Thiadiazoline derivatives for treating cancer KYOWA HAKKO KIRIN CO LTD (JP) 2012-03-21 EP disclosed
EP-1847534-B1 Thiadiazoline derivatives for treating cancer KYOWA HAKKO KIRIN CO LTD (JP) 2011-06-22 EP disclosed
CN-1972919-A Method for producing 4-(benzimidazolylmethylamino)-benzamidines BOEHRINGER INGELHEIM INT (DE) 2007-05-30 CN disclosed