SCHEMBL7587029

SCHEMBL7587029

CCOC(=O)CC(=O)NCCCc1ccc2c(n1)NCCC2

nearest known ligand 0.61

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 16/20 0.61
ITGB3 P05106 13/20 0.61
ITGB6 P18564 9/20 0.50
ITGB5 P18084 6/20 0.50
ITGB8 P26012 6/20 0.50
CXCR4 P61073 3/20 0.50
CCR2 P41597 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22029454 0.87 ITGAV (0.75) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL23542450 0.85 ITGAV (0.52) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL7549076 0.85 ITGB3 (0.74) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL6265738 0.85 ITGAV (0.56) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL19809630 0.84 ITGAV (0.61) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL13720083 0.84 ITGAV (0.69) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL20480976 0.83 ITGAV (0.52) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL22223353 0.83 ITGAV (0.60) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL16607379 0.83 ITGAV (0.60) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL7015442 0.83 ITGB3 (0.68) ITGAVITGB3ITGB6ITGB5ITGB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946165-A4 INTEGRIN ANTAGONISTS MERCK & CO INC (US) 2001-04-11 EP disclosed
EP-0946165-A1 INTEGRIN ANTAGONISTS Merck & Co., Inc. (US) 1999-10-06 EP disclosed
WO-1998018460-A1 INTEGRIN ANTAGONISTS MERCK & CO., INC. (US) 1998-05-07 WO disclosed