SCHEMBL7587185

SCHEMBL7587185

CC#CC(C)(C)c1ccc(OC)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA7 P43166 2/20 0.46
CA9 Q16790 2/20 0.46
CA12 O43570 1/20 0.46
CA14 Q9ULX7 1/20 0.46
TDP1 Q9NUW8 4/20 0.43
MAPK1 P28482 3/20 0.43
ALDH1A1 P00352 3/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 2/20 0.41
RECQL P46063 2/20 0.40
LMNA P02545 1/20 0.40
ALOX15 P16050 1/20 0.40
APEX1 P27695 1/20 0.40
HSD17B10 Q99714 1/20 0.40
AOC3 Q16853 1/20 0.40
APP P05067 1/20 0.39
ACHE P22303 1/20 0.39
KIF11 P52732 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7138584 0.80 CA1 (0.42) CA1CA2CA7CA9CA12
SCHEMBL7591916 0.79 CA1 (0.41) CA1CA2CA7CA9CA12
SCHEMBL26394798 0.79 TRPV1 (0.42) TDP1ALDH1A1CYP3A4MAPTALOX15
SCHEMBL989065 0.77 CA1 (0.48) CA1CA2CA7CA9CA12
SCHEMBL3742483 0.77 CA1 (0.48) CA1CA2CA7CA9CA12
SCHEMBL7592148 0.77 CA1 (0.48) CA1CA2CA7CA9CA12
SCHEMBL7586236 0.76 MEN1 (0.44) CA1CA2CA7CA9CA12
SCHEMBL20936575 0.76 TSHR (0.50) CA1CA2CA7CA9TDP1
SCHEMBL7586544 0.74 LMNA (0.51) CA1CA2TDP1MAPK1ALDH1A1
SCHEMBL24278471 0.74 RAB9A (0.36) MAPK1ALDH1A1MAPTACHEKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780375-B1 3-((5-substituted benzyl)amino)-2-phenylpiperidines as substance p antagonists PFIZER (US) 2002-09-11 EP disclosed
US-5789423-A ANTIALLERGENS, ANTIINFLAMMATORY AGENTS; GASTROINTESTINAL AND CENTRAL NERVOUS SYSTEM DISORDERS PFIZER INC. (US) 1998-08-04 US disclosed
EP-0780375-A1 3-((5-substituted benzyl)amino)-2-phenylpiperidines as substance p antagonists PFIZER INC. (US) 1997-06-25 EP disclosed