SCHEMBL7587674

SCHEMBL7587674

O=C(Nc1nc2ccccc2n1-c1ncccn1)c1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.64
NPC1 O15118 4/20 0.64
KDM4E B2RXH2 7/20 0.59
NPSR1 Q6W5P4 3/20 0.59
TDP1 Q9NUW8 1/20 0.59
MEN1 O00255 4/20 0.56
KMT2A Q03164 4/20 0.56
TSHR P16473 3/20 0.56
TP53 P04637 3/20 0.54
HSD17B10 Q99714 3/20 0.54
USP2 O75604 2/20 0.54
LMNA P02545 1/20 0.54
PDE11A Q9HCR9 1/20 0.54
PDE10A Q9Y233 1/20 0.54
ALDH1A1 P00352 4/20 0.53
SMN1; SMN2 Q16637 3/20 0.53
ADORA3 P0DMS8 3/20 0.51
ADORA2A P29274 1/20 0.51
ADORA1 P30542 1/20 0.51
EGFR P00533 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11707540 0.85 RAB9A (0.69) RAB9ANPC1KDM4ENPSR1TDP1
SCHEMBL7591224 0.80 KDM4E (0.52) RAB9ANPC1KDM4ENPSR1TDP1
SCHEMBL11702096 0.79 RAB9A (0.65) RAB9ANPC1KDM4ENPSR1TDP1
SCHEMBL29510945 0.79 RAB9A (1.00) RAB9ANPC1KDM4ENPSR1TDP1
SCHEMBL14773948 0.79 RAB9A (1.00) RAB9ANPC1KDM4ENPSR1TDP1
SCHEMBL7590440 0.77 BRD4 (0.45) RAB9ANPC1KDM4EMEN1KMT2A
SCHEMBL5089620 0.76 RAB9A (0.70) RAB9ANPC1KDM4ENPSR1TDP1
SCHEMBL11703407 0.76 RAB9A (0.69) RAB9ANPC1KDM4ENPSR1TDP1
SCHEMBL11705615 0.75 RAB9A (0.72) RAB9ANPC1KDM4ENPSR1TDP1
SCHEMBL17916715 0.74 RAB9A (0.89) RAB9ANPC1KDM4ENPSR1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1206260-A4 SRC KINASE INHIBITOR COMPOUNDS MERCK & CO INC (US) 2002-10-30 EP disclosed
EP-1206260-A1 SRC KINASE INHIBITOR COMPOUNDS Merck & Co., Inc. (US) 2002-05-22 EP disclosed
WO-2001000207-A1 SRC KINASE INHIBITOR COMPOUNDS MERCK & CO., INC. (US) 2001-01-04 WO disclosed