SCHEMBL7588677

SCHEMBL7588677

O=C(O)c1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)c(I)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
ALOX15 P16050 3/20 0.37
KDM4E B2RXH2 3/20 0.37
TSHR P16473 1/20 0.37
ACMSD Q8TDX5 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
MGAM O43451 1/20 0.35
LMNA P02545 1/20 0.34
NAPRT Q6XQN6 1/20 0.34
P4HTM Q9NXG6 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ALDH1A1 P00352 6/20 0.34
HSD17B10 Q99714 2/20 0.34
HPGD P15428 1/20 0.34
CYP1A2 P05177 1/20 0.32
MAPT P10636 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PTGER1 P34995 1/20 0.32
GNE Q9Y223 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8023190 0.84 ALDH1A1 (0.39) KDM4ETSHRALDH1A1HSD17B10HPGD
SCHEMBL10917086 0.81 PTGS1 (0.41) PTGS1PTGS2ALOX15KDM4ETSHR
SCHEMBL3038938 0.77 PTGS1 (0.39) PTGS1PTGS2ALOX15KDM4ETSHR
SCHEMBL1423935 0.75 CYP11B1 (0.33) CYP11B1CYP11B2
SCHEMBL8006029 0.74 P2RX7 (0.37) CYP11B1CYP11B2
SCHEMBL8022922 0.74 NOTUM (0.36) L3MBTL1CYP11B1CYP11B2
SCHEMBL6105313 0.70 ALDH1A1 (0.36) PTGS1PTGS2KDM4ETSHRLMNA
SCHEMBL10919181 0.69 BRD4 (0.40) ALDH1A1HPGD
SCHEMBL2720194 0.67 NPC1 (0.34) PTGS2ALOX15KDM4ETDP1ALDH1A1
SCHEMBL23704608 0.67 AKT1 (0.39) ALOX15KDM4ETSHRTDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0904271-A4 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES UNIV PRINCETON (US) 2002-01-23 EP disclosed
US-6066639-A ANTITUMOR AGENTS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2000-05-23 US disclosed
EP-0904271-A1 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1999-03-31 EP disclosed
WO-1997041115-A1 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1997-11-06 WO disclosed