SCHEMBL7589227

SCHEMBL7589227

Nc1cc(N)cc(C(O)CO)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.38
TSHR P16473 2/20 0.38
SCN9A Q15858 3/20 0.35
PLAU P00749 1/20 0.33
LMNA P02545 3/20 0.32
ADRB2 P07550 3/20 0.32
ADRB1 P08588 2/20 0.32
ADRA1A P35348 2/20 0.32
HTR1A P08908 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
OPRK1 P41145 1/20 0.32
SLC6A3 Q01959 1/20 0.32
KDM4E B2RXH2 2/20 0.32
MAPT P10636 2/20 0.31
HPGD P15428 2/20 0.31
APEX1 P27695 2/20 0.31
RECQL P46063 2/20 0.31
BLM P54132 2/20 0.31
TDP1 Q9NUW8 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8417955 0.81 CYP3A4 (0.33) CYP3A4TSHR
SCHEMBL8417924 0.80 SMN1; SMN2 (0.44) CYP3A4TSHRMAPTHPGDMEN1
SCHEMBL18434948 0.77 CYP19A1 (0.46) CYP3A4TSHRPLAUKDM4EMAPT
SCHEMBL10714160 0.77 CYP19A1 (0.46) CYP3A4TSHRPLAUKDM4EMAPT
SCHEMBL2238144 0.77 CPN1 (0.49) CYP3A4TSHRLMNAADRB2ADRB1
SCHEMBL9152377 0.77 CPN1 (0.49) CYP3A4TSHRLMNAADRB2ADRB1
SCHEMBL28252277 0.75 ABCB11 (0.40) TSHRADRB2HPGDTDP1
SCHEMBL207218 0.73 TSHR (0.39) CYP3A4TSHRSCN9ALMNAADRB2
SCHEMBL28919999 0.72 CES2 (0.43) CYP3A4TSHRSCN9AADRB1SLC6A2
SCHEMBL19556861 0.71 CYP3A4 (0.35) CYP3A4TSHRMAPTRECQLTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6448442-B1 X-RAY CONTRAST AGENTS; LOW VISCOSITY IODINATED ARYL COMPOUNDS AMERSHAM HEALTH AS (NO) 2002-09-10 US disclosed
US-6310243-B1 BENZENE COMPOUNDS IN WHICH 3 NON-ADJACENT RING ATOMS ARE SUBSTITUTED WITH IODINE, 2 OF THE REMAINING RING ATOMS ARE AMIDE SUBSTITUTED WITH HYDROXY AND THE OTHER REMAINING RING ATOM IS A NON-AMIDE, HYDROXY-SUBSTITUTED NONIONIC MOIETY NYCOMED IMAGING AS (NO) 2001-10-30 US disclosed
US-5993780-A A POLYIODOARYLALKYL ALCOHOL OR DERIVATIVE NYCOMED IMAGING AS (NO) 1999-11-30 US disclosed
US-5882628-A Contrast media NYCOMED IMAGING AS (NO) 1999-03-16 US disclosed
EP-0782564-A1 IODINATED X-RAY CONTRAST MEDIA NYCOMED IMAGING AS (NO) 1997-07-09 EP disclosed
WO-1996009282-A1 IODINATED X-RAY CONTRAST MEDIA NYCOMED IMAGING A/S (NO) 1996-03-28 WO disclosed