SCHEMBL7590648

SCHEMBL7590648

O=C(O)C[C@@H](c1nc2ccccc2o1)N1CCN(CCCC2=CC=C3CCCNC3N2)C1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 11/20 0.43
ITGB3 P05106 9/20 0.43
ITGB8 P26012 6/20 0.39
ITGB6 P18564 5/20 0.39
ITGA5 P08648 4/20 0.38
ITGB1 P05556 1/20 0.38
ITGA2B P08514 1/20 0.38
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC9 Q9UKV0 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
DRD2 P14416 1/20 0.31
DRD4 P21917 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7590552 1.00 ITGAV (0.43) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7557082 1.00 ITGAV (0.43) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7555650 0.85 ITGB8 (0.44) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7594404 0.85 ITGB8 (0.44) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7596620 0.85 ITGB8 (0.44) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL4374458 0.85 ITGB3 (0.45) ITGAVITGB3ITGB1ITGA2BHDAC3
SCHEMBL7591361 0.84 ITGAV (0.47) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7589610 0.84 ITGAV (0.47) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7589125 0.82 ITGAV (0.61) ITGAVITGB3ITGB8ITGB6ITGA5
SCHEMBL7591261 0.82 ITGAV (0.61) ITGAVITGB3ITGB8ITGB6ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040111-A1 INTEGRIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2000-10-04 EP disclosed
WO-1999031099-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO disclosed