SCHEMBL7593239

SCHEMBL7593239

CCCN1C(=O)C(N(C(N)=O)c2nnc(C)s2)N=C(N2CCN(C)CC2)c2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 12/20 0.51
BDKRB1 P46663 6/20 0.36
NOTCH1 P46531 1/20 0.35
RBPJ Q06330 1/20 0.35
DRD2 P14416 1/20 0.34
DRD1 P21728 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9566076 0.83 CCKBR (0.49) CCKBRBDKRB1NOTCH1RBPJDRD2
SCHEMBL7594182 0.77 CCKBR (0.70) CCKBRBDKRB1
SCHEMBL9368725 0.74 CCKBR (0.49) CCKBRDRD2
SCHEMBL8540989 0.74 CCKBR (0.55) CCKBRDRD2DRD1
Acetic Acid SCHEMBL8883854 0.73 CCKBR (0.56) CCKBRBDKRB1NOTCH1RBPJDRD2
Trifluoroacetic Acid SCHEMBL8590781 0.70 CCKBR (0.56) CCKBRBDKRB1NOTCH1RBPJDRD2
Benzene SCHEMBL8824680 0.70 CCKBR (0.64) CCKBRBDKRB1NOTCH1RBPJ
SCHEMBL9369254 0.67 CCKBR (0.73) CCKBRBDKRB1
SCHEMBL9368456 0.67 CCKBR (1.00) CCKBR
SCHEMBL9368848 0.67 CCKBR (1.00) CCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002099388-A2 BENZODIAZEPINE BRADYKININ ANTAGONISTS MERCK & CO., INC. (US) 2002-12-12 WO claimed