SCHEMBL9566076

SCHEMBL9566076

CCCN1C(=O)[C@@H](N(C(N)=O)c2ccc(N(C)C)cc2)N=C(N2CCN(C)CC2)c2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 9/20 0.49
BDKRB1 P46663 5/20 0.37
DRD2 P14416 4/20 0.36
DRD1 P21728 2/20 0.36
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
PKM P14618 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
NOTCH1 P46531 1/20 0.35
RBPJ Q06330 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7593239 0.83 CCKBR (0.51) CCKBRBDKRB1DRD2DRD1NOTCH1
SCHEMBL9368725 0.82 CCKBR (0.49) CCKBRDRD2
SCHEMBL9369254 0.78 CCKBR (0.73) CCKBRBDKRB1
SCHEMBL8540989 0.76 CCKBR (0.55) CCKBRDRD2DRD1MEN1ALDH1A1
Acetic Acid SCHEMBL8883854 0.76 CCKBR (0.56) CCKBRBDKRB1DRD2DRD1ALDH1A1
SCHEMBL7597644 0.75 BDKRB1 (0.39) CCKBRBDKRB1KDM4EALDH1A1MAPT
SCHEMBL7592838 0.74 BDKRB1 (0.55) CCKBRBDKRB1
SCHEMBL9008723 0.73 BDKRB1 (0.54) CCKBRBDKRB1
Trifluoroacetic Acid SCHEMBL8590781 0.73 CCKBR (0.56) CCKBRBDKRB1DRD2DRD1NOTCH1
SCHEMBL9368479 0.73 CCKBR (0.81) CCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0539170-A1 Benzodiazepine derivatives and their use as antagonists of cholecystokinin and/or gastrin receptors MERCK SHARP & DOHME LTD. (GB) 1993-04-28 EP disclosed