SCHEMBL7598348

SCHEMBL7598348

COC(=O)C(Cc1cnc[nH]1)NC(=O)O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 3/20 0.55
ICAM1 P05362 3/20 0.55
ITGAL P20701 3/20 0.55
HTR1D P28221 2/20 0.51
HTR2C P28335 2/20 0.51
HTR1E P28566 2/20 0.51
HTR2B P41595 2/20 0.51
HTR2A P28223 1/20 0.51
HTR3A P46098 1/20 0.51
CYP3A4 P08684 3/20 0.50
SLC7A5 Q01650 1/20 0.50
ALOX5 P09917 1/20 0.48
PDCD1 Q15116 1/20 0.47
CD274 Q9NZQ7 1/20 0.47
SLC6A5 Q9Y345 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
ALDH1A1 P00352 2/20 0.45
GABRA1 P14867 1/20 0.45
TSHR P16473 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5808674 0.89 HTR1D (0.51) ITGB2ICAM1ITGALHTR1DHTR2C
SCHEMBL13912236 0.86 HTR1D (0.49) ITGB2ICAM1ITGALHTR1DHTR2C
SCHEMBL19051483 0.85 SLC6A5 (0.53) ITGB2ICAM1ITGALHTR1DHTR2C
SCHEMBL13897023 0.85 CYP3A4 (0.49) ITGB2ICAM1ITGALHTR1DHTR2C
SCHEMBL10664287 0.85 CYP3A4 (0.49) ITGB2ICAM1ITGALHTR1DHTR2C
SCHEMBL27413426 0.85 ITGB2 (0.67) ITGB2ICAM1ITGALCYP3A4SLC7A5
SCHEMBL29002721 0.85 HTR1D (0.48) ITGB2ICAM1ITGALHTR1DHTR2C
SCHEMBL28221477 0.84 HRH3 (0.53) ITGB2ICAM1ITGALSLC6A5
SCHEMBL11158707 0.84 ITGB2 (0.58) ITGB2ICAM1ITGALHTR1DHTR2C
SCHEMBL23901492 0.84 CYP3A4 (0.48) ITGB2ICAM1ITGALHTR1DHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1266900-A1 Carbamates of rapamycin Wyeth (US) 2002-12-18 EP disclosed
US-5411967-A Antiinflammatory, immunosuppressant, antitumor AMERICAN HOME PRODUCTS CORPORATION (US) 1995-05-02 US disclosed
EP-0593227-A1 Carbamates of rapamycin AMERICAN HOME PRODUCTS CORPORATION (US) 1994-04-20 EP disclosed
US-5302584-A Immunosuppressants AMERICAN HOME PRODUCTS CORPORATION (US) 1994-04-12 US disclosed