SCHEMBL7598524

SCHEMBL7598524

CC(=O)OCc1cc(CBr)cc(C(=O)O)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
IDH1 O75874 1/20 0.40
CYP3A4 P08684 1/20 0.40
PKM P14618 3/20 0.37
CA12 O43570 2/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA7 P43166 2/20 0.37
CA9 Q16790 2/20 0.37
CA14 Q9ULX7 2/20 0.37
CA3 P07451 1/20 0.37
CA4 P22748 1/20 0.37
CA6 P23280 1/20 0.37
CA5A P35218 1/20 0.37
CA5B Q9Y2D0 1/20 0.37
MRGPRX4 Q96LA9 6/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PTGS2 P35354 1/20 0.35
TSHR P16473 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2226759 0.82 TTR (0.44) ALDH1A1PKMCA12CA1CA2
SCHEMBL7593857 0.80 MRGPRX4 (0.40) ALDH1A1PKMCA12CA1CA2
Acetic Acid SCHEMBL28155950 0.80 TPMT (0.43) ALDH1A1PKMCA12CA1CA2
SCHEMBL5666942 0.80 ALDH1A1 (0.64) ALDH1A1IDH1CYP3A4CA2RAB9A
SCHEMBL5351634 0.79 ALDH1A1 (0.43) ALDH1A1IDH1CYP3A4CA2MEN1
SCHEMBL1866724 0.78 TTR (0.44) ALDH1A1PKMCA12CA1CA2
SCHEMBL7594237 0.76 PKM (0.38) ALDH1A1PKMCA12CA1CA2
SCHEMBL31160231 0.76 ALDH1A1 (0.61) ALDH1A1IDH1CYP3A4CA2RAB9A
SCHEMBL990642 0.76 ALDH1A1 (0.61) ALDH1A1IDH1CYP3A4CA2RAB9A
SCHEMBL1792464 0.75 KMT2A (0.46) ALDH1A1IDH1MRGPRX4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000038-B1 NOVEL PYRIMIDIN DERIVATIVES ASTRAZENECA AB (SE) 2002-11-06 EP disclosed
US-6200981-B1 FOR TREATING INFLAMMATORY DISEASES SUCH AS ASTHMA, INFLAMMATORY BOWEL DISEASE, PSORIASIS, RHEUMATOID ARTHRITIS, MYOCARDIAL ISCHAEMIA, CYSTIC FIBROSIS, ARTHEREOSCLEROSIS, RESTENOSIS, PERIDONTAL DISEASE, SEPTIC SHOCK, OSTEOARTHRITIS ASTRAZENECA UK LIMITED (GB) 2001-03-13 US disclosed