SCHEMBL7599559

SCHEMBL7599559

O=C(O)Nc1nccc2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FDPS P14324 1/20 0.54
DRD2 P14416 1/20 0.50
DRD4 P21917 1/20 0.50
DRD3 P35462 1/20 0.50
RAB9A P51151 2/20 0.49
CYP2A6 P11509 1/20 0.48
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
HPGD P15428 1/20 0.48
MAP3K7 O43318 2/20 0.46
MAP3K6 O95382 2/20 0.46
MAP3K5 Q99683 2/20 0.46
CNR2 P34972 1/20 0.46
ADORA3 P0DMS8 2/20 0.44
NPC1 O15118 1/20 0.44
POLB P06746 1/20 0.44
KMT2A Q03164 1/20 0.44
F12 P00748 1/20 0.44
PLAU P00749 1/20 0.44
NCF1 P14598 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29825764 1.00 FDPS (0.54) FDPSDRD2DRD4DRD3RAB9A
SCHEMBL5380631 0.86 FDPS (0.51) FDPSDRD2DRD4DRD3RAB9A
SCHEMBL5874038 0.85 ADORA3 (0.62) FDPSRAB9ACNR2ADORA3NPC1
SCHEMBL4411955 0.84 FDPS (0.53) FDPSDRD2DRD4DRD3RAB9A
SCHEMBL10051128 0.84 FDPS (0.53) FDPSDRD2DRD4DRD3RAB9A
SCHEMBL2361181 0.84 KDM4E (0.56) FDPSDRD2DRD4DRD3RAB9A
SCHEMBL13685315 0.81 TRPV1 (0.49) FDPSDRD2DRD4DRD3RAB9A
SCHEMBL4410540 0.80 KMT2A (0.50) FDPSDRD2DRD4DRD3RAB9A
SCHEMBL7937683 0.80 FDPS (0.49) FDPSDRD2DRD4DRD3RAB9A
SCHEMBL31606592 0.80 KMT2A (0.50) FDPSDRD2DRD4DRD3RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106257976-A Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2016-12-28 CN disclosed
EP-1266900-A1 Carbamates of rapamycin Wyeth (US) 2002-12-18 EP disclosed
US-5411967-A Antiinflammatory, immunosuppressant, antitumor AMERICAN HOME PRODUCTS CORPORATION (US) 1995-05-02 US disclosed
CN-1091135-A The carbamate of Wyeth-Ayerst Laboratories AMERICAN HOME PROD (US) 1994-08-24 CN disclosed
EP-0593227-A1 Carbamates of rapamycin AMERICAN HOME PRODUCTS CORPORATION (US) 1994-04-20 EP disclosed
US-5302584-A Immunosuppressants AMERICAN HOME PRODUCTS CORPORATION (US) 1994-04-12 US disclosed