SCHEMBL7601887

SCHEMBL7601887

Cc1ccccc1C(C)c1ccc(Cl)nn1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.46
GAA P10253 5/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
ESR1 P03372 1/20 0.37
LMNA P02545 5/20 0.37
KDM4E B2RXH2 1/20 0.37
KMT2A Q03164 1/20 0.36
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
CTSA P10619 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27446618 0.79 ALDH1A1 (0.43) ALDH1A1GAAL3MBTL1LMNAKMT2A
SCHEMBL23879238 0.78 ALDH1A1 (0.73) ALDH1A1GAAL3MBTL1ESR1LMNA
SCHEMBL30452159 0.78 ALDH1A1 (0.73) ALDH1A1GAAL3MBTL1ESR1LMNA
SCHEMBL23879259 0.76 GAA (0.43) ALDH1A1GAAL3MBTL1LMNAKDM4E
SCHEMBL30452188 0.76 GAA (0.43) ALDH1A1GAAL3MBTL1LMNAKDM4E
SCHEMBL146510 0.72 ESR1 (0.56) ALDH1A1GAAESR1ADRA2AADRA2B
SCHEMBL2600116 0.71 ALDH1A1 (0.46) ALDH1A1GAAL3MBTL1LMNAKMT2A
SCHEMBL28752820 0.69 SLC6A2 (0.42) ALDH1A1GAAL3MBTL1ESR1LMNA
SCHEMBL31405028 0.69 ALDH1A1 (0.44) ALDH1A1GAAL3MBTL1LMNAKMT2A
SCHEMBL8505132 0.68 ADRA2A (0.37) ALDH1A1GAAESR1LMNAADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810218-B1 6-Benzyl-2H-pyridazin-3-one derivatives,their preparation and their use as inhibitors of prostaglandin G/H synthase I and II (COX I and COX II) HOFFMANN LA ROCHE (CH) 2002-12-04 EP disclosed
EP-0810218-A1 6-Benzyl-2H-pyridazin-3-one derivatives,their preparation and their use as inhibitors of prostaglandin G/H synthase I and II (COX I and COX II) F. HOFFMANN-LA ROCHE AG (CH) 1997-12-03 EP disclosed