SCHEMBL7603493

SCHEMBL7603493

COc1cccc(C(N)CCOc2cc(Cl)c(F)cc2C(N)=O)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.39
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
TYK2 P29597 1/20 0.39
JAK3 P52333 1/20 0.39
NNMT P40261 1/20 0.37
LMNA P02545 1/20 0.36
PARP10 Q53GL7 2/20 0.36
PARP15 Q460N3 1/20 0.36
PARP14 Q460N5 1/20 0.36
HTR1A P08908 1/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
SLC6A3 Q01959 2/20 0.36
RPS6KB1 P23443 2/20 0.36
KCNH2 Q12809 1/20 0.36
CSF1R P07333 3/20 0.35
ROCK2 O75116 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6492057 0.82 CYP2D6 (0.43) HTTJAK2JAK1TYK2JAK3
SCHEMBL6983849 0.81 CYP2D6 (0.44) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
Oxalic Acid SCHEMBL6553236 0.80 CYP2D6 (0.47) HTTJAK2JAK1TYK2JAK3
Oxalic Acid SCHEMBL6493248 0.67 NOS2 (0.67) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL6498984 0.65 NOS2 (0.62) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL1439439 0.65 PDCD1LG2 (0.42) NNMTCYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL1439436 0.65 PDCD1LG2 (0.42) NNMTCYP3A4CYP2D6SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL18765506 0.64 PDCD1LG2 (0.41) NNMTCYP3A4CYP2D6SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL18765505 0.64 PDCD1LG2 (0.41) NNMTCYP3A4CYP2D6SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL29676921 0.64 PDCD1LG2 (0.41) NNMTCYP3A4CYP2D6SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1263711-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES AstraZeneca AB (SE) 2002-12-11 EP disclosed
WO-2001062704-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES ASTRAZENECA AB (SE) 2001-08-30 WO disclosed