SCHEMBL6983849

SCHEMBL6983849

COc1cccc(C(N)CCOc2cc(Cl)c(F)cc2C#N)n1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.44
SLC6A2 P23975 4/20 0.44
SLC6A4 P31645 4/20 0.44
NOS2 P35228 2/20 0.44
MRGPRX4 Q96LA9 1/20 0.38
CYP3A4 P08684 3/20 0.34
SLC6A3 Q01959 2/20 0.34
KCNH2 Q12809 1/20 0.34
SLC22A12 Q96S37 2/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
F11 P03951 2/20 0.34
S1PR1 P21453 2/20 0.33
EGFR P00533 2/20 0.33
S1PR3 Q99500 1/20 0.33
AAK1 Q2M2I8 1/20 0.33
APLNR P35414 2/20 0.33
TRPV4 Q9HBA0 1/20 0.33
ERBB2 P04626 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6498984 0.82 NOS2 (0.62) CYP2D6SLC6A2SLC6A4NOS2MRGPRX4
SCHEMBL7603493 0.81 HTT (0.39) CYP2D6SLC6A2SLC6A4CYP3A4SLC6A3
Oxalic Acid SCHEMBL6493248 0.78 NOS2 (0.67) CYP2D6SLC6A2SLC6A4NOS2MRGPRX4
SCHEMBL6981893 0.74 NOS2 (0.52) CYP2D6SLC6A2SLC6A4NOS2MRGPRX4
SCHEMBL7601784 0.70 CYP2D6 (0.44) CYP2D6SLC6A2SLC6A4NOS2MRGPRX4
SCHEMBL6980102 0.70 CYP2D6 (0.43) CYP2D6SLC6A2SLC6A4NOS2MRGPRX4
SCHEMBL21691198 0.68 CYP2D6 (0.48) CYP2D6SLC6A2SLC6A4NOS2S1PR1
SCHEMBL31376036 0.68 CYP2D6 (0.48) CYP2D6SLC6A2SLC6A4NOS2S1PR1
SCHEMBL7599969 0.67 CYP2D6 (0.46) CYP2D6SLC6A2SLC6A4NOS2SLC22A12
SCHEMBL1695992 0.67 MRGPRX4 (0.47) CYP2D6SLC6A2SLC6A4NOS2MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003523988-A 2003-08-12 JP claimed
EP-1263711-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES AstraZeneca AB (SE) 2002-12-11 EP claimed
WO-2001062704-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES ASTRAZENECA AB (SE) 2001-08-30 WO claimed
EP-1263711-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES AstraZeneca AB (SE) 2002-12-11 EP disclosed
WO-2001062704-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES ASTRAZENECA AB (SE) 2001-08-30 WO disclosed