SCHEMBL7603978

SCHEMBL7603978

O=CC(Br)c1cccc2c1-c1ccccc1C2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.40
POLB P06746 1/20 0.38
HTR2B P41595 1/20 0.38
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35
RRM1 P23921 1/20 0.35
RRM2B Q7LG56 1/20 0.35
BCHE P06276 1/20 0.34
CES1 P23141 1/20 0.34
MAPK8 P45983 1/20 0.33
MAPK9 P45984 1/20 0.33
MAPK10 P53779 1/20 0.33
MIF P14174 3/20 0.33
CYP3A4 P08684 2/20 0.33
HSD17B10 Q99714 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
MAP3K9 P80192 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19682354 0.78 CYP1A2 (0.41) MAOAPOLBHTR2BCHRM2CHRM1
SCHEMBL22310126 0.74 HTR2B (0.43) MAOAPOLBHTR2BBCHECES1
SCHEMBL8160473 0.74 MAOA (0.42) MAOAPOLBHTR2BCHRM2CHRM1
SCHEMBL26461857 0.71 HTR2B (0.44) MAOAPOLBHTR2BCHRM2CHRM1
SCHEMBL28167254 0.71 POLB (0.41) MAOAPOLBHTR2BBCHECES1
SCHEMBL1626146 0.71 MAOA (0.52) MAOAPOLBHTR2BBCHECES1
SCHEMBL2120191 0.70 MAOA (0.47) MAOAPOLBHTR2BBCHECES1
SCHEMBL28004757 0.70 MAOA (0.54) MAOAPOLBHTR2BBCHECES1
Fluorene SCHEMBL28167258 0.70 HTR2B (0.40) MAOAPOLBHTR2BBCHECES1
SCHEMBL28004759 0.68 MAOA (0.52) MAOAPOLBHTR2BCHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1252163-A2 4-PYRIDYL-AND 2,4-PYRIMIDINYL-SUBSTITUTED PYRROLE DERIVATIVES AND THEIR USE IN PHARMACY MERCKLE GMBH (DE) 2002-10-30 EP disclosed
WO-2001057042-A2 4-PYRIDYL-AND 2,4-PYRIMIDINYL-SUBSTITUTED PYRROLE DERIVATIVES AND THEIR USE IN PHARMACY MERCKLE GMBH (DE) 2001-08-09 WO disclosed