SCHEMBL7604748

SCHEMBL7604748

CCOC(=O)CCCc1ccc(OCC2CO2)c(C#N)c1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 3/20 0.48
CASR P41180 3/20 0.44
CYP2D6 P10635 3/20 0.44
ADRB2 P07550 2/20 0.44
SLC6A2 P23975 2/20 0.44
SLC6A4 P31645 2/20 0.44
SLC6A3 Q01959 2/20 0.44
KCNH2 Q12809 2/20 0.44
S1PR1 P21453 2/20 0.41
CYP4Z1 Q86W10 1/20 0.39
CYP4F11 Q9HBI6 1/20 0.39
CYP4F12 Q9HCS2 1/20 0.39
TNF P01375 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7604752 1.00 MGLL (0.48) MGLLCASRCYP2D6ADRB2SLC6A2
SCHEMBL7604097 0.94 MGLL (0.48) MGLLCASRCYP2D6ADRB2SLC6A2
SCHEMBL7604094 0.94 MGLL (0.48) MGLLCASRCYP2D6ADRB2SLC6A2
SCHEMBL6374360 0.94 CASR (0.49) MGLLCASRCYP2D6ADRB2SLC6A2
SCHEMBL7603924 0.87 CASR (0.52) MGLLCASRCYP2D6ADRB2SLC6A2
SCHEMBL7603925 0.87 CASR (0.52) MGLLCASRCYP2D6ADRB2SLC6A2
SCHEMBL11023521 0.85 MGLL (0.50) MGLLCYP4Z1CYP4F11CYP4F12
SCHEMBL11023146 0.80 MGLL (0.59) MGLLCYP4Z1CYP4F11CYP4F12
SCHEMBL11021493 0.78 CYP4F2 (0.45) MGLLCYP4Z1
SCHEMBL11020005 0.78 CYP4F2 (0.45) MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6395919-B1 Calcilytic compounds SMITHKLINE BEECHAM CORPORATION 2002-05-28 US disclosed
EP-1070048-A4 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2001-11-07 EP disclosed
EP-1070048-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2001-01-24 EP disclosed
WO-1999051569-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1999-10-14 WO disclosed