SCHEMBL7604891

SCHEMBL7604891

CC(O)c1ccc(N)c([N+](=O)[O-])c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.56
TDP1 Q9NUW8 4/20 0.55
MAPT P10636 4/20 0.55
ALDH1A1 P00352 3/20 0.55
MEN1 O00255 3/20 0.55
KMT2A Q03164 3/20 0.55
POLB P06746 2/20 0.55
CYP3A4 P08684 1/20 0.55
ALOX15 P16050 1/20 0.55
ADRB2 P07550 1/20 0.55
LMNA P02545 1/20 0.51
PKM P14618 1/20 0.47
EPAS1 Q99814 1/20 0.47
CRHBP P24387 1/20 0.45
CRHR2 Q13324 1/20 0.45
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
APP P05067 1/20 0.42
GPR35 Q9HC97 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL978898 0.86 TSHR (0.59) TSHRTDP1MAPTALDH1A1MEN1
SCHEMBL28135866 0.83 TSHR (0.53) TSHRTDP1MAPTALDH1A1MEN1
SCHEMBL20362349 0.83 TSHR (0.56) TSHRTDP1MAPTALDH1A1MEN1
SCHEMBL4136656 0.82 LMNA (0.55) TSHRTDP1MAPTALDH1A1MEN1
SCHEMBL11462352 0.82 TSHR (0.51) TSHRTDP1MAPTALDH1A1MEN1
SCHEMBL15887336 0.82 TSHR (0.51) TSHRTDP1MAPTALDH1A1MEN1
SCHEMBL4434685 0.81 ALDH1A1 (0.53) TSHRTDP1MAPTALDH1A1MEN1
SCHEMBL15762737 0.81 EPAS1 (0.48) TSHRMAPTALDH1A1MEN1KMT2A
SCHEMBL10438572 0.80 TSHR (0.53) TSHRTDP1MAPTALDH1A1MEN1
SCHEMBL16654104 0.80 TSHR (0.53) TSHRTDP1MAPTALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1212096-A2 DRUG CONJUGATES AND METHODS OF DESIGNING THE SAME Brenner, Sydney (US) 2002-06-12 EP disclosed
WO-2001013958-A2 DRUG CONJUGATES AND METHODS OF DESIGNING THE SAME BRENNER SYDNEY (US) 2001-03-01 WO disclosed