SCHEMBL7604955

SCHEMBL7604955

COc1cccc2c1C(=O)OC(=O)C2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 2/20 0.43
CA12 O43570 1/20 0.43
TOP1 P11387 1/20 0.43
ALDH1A1 P00352 6/20 0.41
KDM4E B2RXH2 5/20 0.41
MAPT P10636 5/20 0.41
HPGD P15428 4/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 4/20 0.40
MEN1 O00255 3/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
ODC1 P11926 1/20 0.40
HTR2A P28223 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4140771 0.82 CA12 (0.54) CA9CA12ALDH1A1KDM4EMAPT
SCHEMBL2340155 0.81 KDM4E (0.62) ALDH1A1KDM4EMAPTHPGDNPC1
SCHEMBL2338034 0.80 KDM4E (0.42) CA9CA12ALDH1A1KDM4EMAPT
SCHEMBL2047592 0.79 TOP1 (0.47) CA9CA12TOP1ALDH1A1KDM4E
SCHEMBL1647356 0.79 MAPT (0.52) CA9TOP1ALDH1A1KDM4EMAPT
SCHEMBL2331538 0.78 GRIA1 (0.38) CA9ALDH1A1KDM4EMAPTHPGD
SCHEMBL349476 0.76 ALDH1A1 (0.50) ALDH1A1KDM4EHPGDSMN1; SMN2CYP1A2
SCHEMBL11124354 0.76 CA12 (0.45) CA9CA12ALDH1A1KDM4EMAPT
SCHEMBL2832148 0.74 TDP2 (0.51) ALDH1A1MAPTCYP1A2CYP3A4KMT2A
SCHEMBL1029836 0.74 KDM4E (0.67) CA9TOP1KDM4EMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020098598-A1 Method for tracking compounds in solution phase combinatorial chemistry NEXUS BIOSYSTEMS, INC. 2002-07-25 US disclosed
US-5399702-A Leukotriene antagonists; antiasthmatic, antiallergen, and antianaphylactic agents HOFFMANN-LA ROCHE INC. (US) 1995-03-21 US disclosed
EP-0577003-A1 Thiazolylvinylphenyl derivatives F. HOFFMANN-LA ROCHE AG (CH) 1994-01-05 EP disclosed
US-5273986-A A substituted phenylalkyleneamidophenyleneethylene thiazole HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed