SCHEMBL7605645

SCHEMBL7605645

O=C(O)c1ccc2c(c1)C(=O)CCCO2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
MAPK1 P28482 1/20 0.49
CTNNB1 P35222 1/20 0.46
WNT3A P56704 1/20 0.46
NPC1 O15118 5/20 0.45
RAB9A P51151 5/20 0.45
HPGD P15428 3/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
TTR P02766 1/20 0.41
TSHR P16473 2/20 0.41
RECQL P46063 1/20 0.41
GRM5 P41594 1/20 0.41
SRD5A2 P31213 1/20 0.41
STAT3 P40763 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6293635 0.90 ALDH1A1 (0.51) ALDH1A1MAPK1NPC1RAB9AHPGD
SCHEMBL2260234 0.84 SMN1; SMN2 (0.46) ALDH1A1MAPK1NPC1RAB9AHPGD
SCHEMBL8016583 0.81 HPGD (0.46) ALDH1A1CTNNB1WNT3ANPC1RAB9A
SCHEMBL31262479 0.80 CTNNB1 (0.67) ALDH1A1MAPK1CTNNB1WNT3ANPC1
SCHEMBL875455 0.80 CTNNB1 (0.67) ALDH1A1MAPK1CTNNB1WNT3ANPC1
SCHEMBL8019602 0.80 MAOA (0.60) ALDH1A1CTNNB1WNT3ARAB9AHPGD
SCHEMBL1429751 0.80 ALDH1A1 (0.55) ALDH1A1MAPK1HPGDKMT2AMEN1
SCHEMBL7605647 0.79 GRM5 (0.49) ALDH1A1CTNNB1WNT3ANPC1RAB9A
SCHEMBL1344385 0.79 AKR1B1 (0.44) ALDH1A1CTNNB1WNT3ARAB9AHPGD
SCHEMBL1533619 0.79 MAOB (0.63) ALDH1A1MAPK1NPC1RAB9AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0922703-B1 Substituted heterocyclic benzocycloalkenes and their use as analgesically active compounds GRUENENTHAL GMBH (DE) 2002-12-04 EP disclosed
US-6013809-A ANALGESICS GRUENENTHAL GMBH (DE) 2000-01-11 US disclosed
EP-0922703-A1 Substituted heterocyclic benzocycloalkenes and their use as analgesically active compounds Grünenthal GmbH (DE) 1999-06-16 EP disclosed