SCHEMBL7605883

SCHEMBL7605883

COC(=O)c1cc(C(O)CN(CCC(c2ccc(OC)cc2)c2ccc(OC)cc2)Cc2ccccc2)ccc1OCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
MAPT P10636 2/20 0.45
NR1H3 Q13133 2/20 0.45
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
NPC1 O15118 2/20 0.43
HTT P42858 2/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
HPGD P15428 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
SLC1A5 Q15758 1/20 0.41
PTPN2 P17706 1/20 0.40
PTPN1 P18031 1/20 0.40
PTPN6 P29350 1/20 0.40
LRRK2 Q5S007 1/20 0.40
F2 P00734 1/20 0.40
F7 P08709 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7606163 0.92 NR1H3 (0.47) ALDH1A1NR1H3MEN1KMT2ANPC1
SCHEMBL7607627 0.85 NR1H3 (0.44) ALDH1A1MAPTNR1H3MEN1KMT2A
SCHEMBL7607631 0.85 NR1H3 (0.44) ALDH1A1MAPTNR1H3MEN1KMT2A
SCHEMBL7606596 0.85 NR1H3 (0.43) ALDH1A1MAPTNR1H3MEN1KMT2A
SCHEMBL7605016 0.83 MAPT (0.43) ALDH1A1MAPTNR1H3MEN1KMT2A
SCHEMBL7606574 0.83 NR1H3 (0.49) ALDH1A1MAPTNR1H3MEN1KMT2A
SCHEMBL7605885 0.82 MAPT (0.45) ALDH1A1MAPTMEN1KMT2ANPC1
SCHEMBL7610085 0.82 HDAC3 (0.44) ALDH1A1MAPTNR1H3MEN1KMT2A
SCHEMBL13708415 0.81 BCHE (0.43) ALDH1A1MAPTMEN1KMT2AHTT
SCHEMBL6320449 0.80 NR1H3 (0.47) ALDH1A1MAPTNR1H3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230210-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-08-14 EP disclosed
WO-2001036375-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-25 WO disclosed