SCHEMBL7605985

SCHEMBL7605985

CCC(CCOc1cc(Cl)c(F)cc1C#N)NCCOC

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 0.40
CYP2D6 P10635 4/20 0.40
SLC6A2 P23975 4/20 0.40
NOS2 P35228 4/20 0.40
BCL2A1 Q16548 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.34
F11 P03951 2/20 0.34
EGFR P00533 2/20 0.32
ERBB2 P04626 2/20 0.32
S1PR1 P21453 1/20 0.32
S1PR3 Q99500 1/20 0.32
SRC P12931 3/20 0.32
AR P10275 1/20 0.31
ALDH1A1 P00352 1/20 0.31
SLC22A12 Q96S37 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6332207 0.76 NOS2 (0.52) SLC6A4CYP2D6SLC6A2NOS2BCL2A1
SCHEMBL7604218 0.72 SLC6A4 (0.41) SLC6A4CYP2D6SLC6A2NOS2BCL2A1
Oxalic Acid SCHEMBL6337578 0.72 CYP2D6 (0.53) SLC6A4CYP2D6SLC6A2NOS2BCL2A1
SCHEMBL6980102 0.70 CYP2D6 (0.43) SLC6A4CYP2D6SLC6A2NOS2BCL2A1
SCHEMBL6329018 0.69 SLC6A4 (0.70) SLC6A4CYP2D6SLC6A2NOS2BCL2A1
SCHEMBL6503271 0.69 SLC6A4 (0.72) SLC6A4CYP2D6SLC6A2NOS2
Hydrochloric Acid SCHEMBL6328545 0.68 SLC6A4 (0.71) SLC6A4CYP2D6SLC6A2NOS2BCL2A1
SCHEMBL21691198 0.68 CYP2D6 (0.48) SLC6A4CYP2D6SLC6A2NOS2BCL2A1
SCHEMBL31376036 0.68 CYP2D6 (0.48) SLC6A4CYP2D6SLC6A2NOS2BCL2A1
Oxalic Acid SCHEMBL7665481 0.67 CYP2D6 (0.42) SLC6A4CYP2D6SLC6A2NOS2BCL2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1263715-A1 NOVEL PHENYLHETEROALKYLAMINE DERIVATIVES AstraZeneca AB (SE) 2002-12-11 EP claimed
WO-2001062714-A1 NOVEL PHENYLHETEROALKYLAMINE DERIVATIVES ASTRAZENECA AB (SE) 2001-08-30 WO claimed
EP-1263715-A1 NOVEL PHENYLHETEROALKYLAMINE DERIVATIVES AstraZeneca AB (SE) 2002-12-11 EP disclosed
WO-2001062714-A1 NOVEL PHENYLHETEROALKYLAMINE DERIVATIVES ASTRAZENECA AB (SE) 2001-08-30 WO disclosed