SCHEMBL6980102

SCHEMBL6980102

CNC(CCOc1cc(Cl)c(F)cc1C#N)c1ncccn1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.43
SLC6A2 P23975 2/20 0.43
SLC6A4 P31645 2/20 0.43
NOS2 P35228 2/20 0.43
S1PR3 Q99500 7/20 0.39
MRGPRX4 Q96LA9 1/20 0.37
S1PR1 P21453 3/20 0.35
SLC22A12 Q96S37 3/20 0.35
F11 P03951 2/20 0.34
BCL2A1 Q16548 1/20 0.34
CYP11B2 P19099 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7599969 0.83 CYP2D6 (0.46) CYP2D6SLC6A2SLC6A4NOS2S1PR3
SCHEMBL7601784 0.82 CYP2D6 (0.44) CYP2D6SLC6A2SLC6A4NOS2S1PR3
SCHEMBL6491537 0.77 SLC6A4 (0.53) CYP2D6SLC6A2SLC6A4NOS2S1PR3
Hydrochloric Acid SCHEMBL6490386 0.76 SLC6A4 (0.53) CYP2D6SLC6A2SLC6A4NOS2S1PR3
SCHEMBL7604218 0.76 SLC6A4 (0.41) CYP2D6SLC6A2SLC6A4NOS2MRGPRX4
SCHEMBL6981893 0.72 NOS2 (0.52) CYP2D6SLC6A2SLC6A4NOS2S1PR3
SCHEMBL7605985 0.70 SLC6A4 (0.40) CYP2D6SLC6A2SLC6A4NOS2S1PR3
SCHEMBL6983849 0.70 CYP2D6 (0.44) CYP2D6SLC6A2SLC6A4NOS2S1PR3
SCHEMBL6577181 0.68 SLC6A4 (0.53) CYP2D6SLC6A2SLC6A4NOS2S1PR3
SCHEMBL6982533 0.67 CYP2D6 (0.43) CYP2D6SLC6A2SLC6A4NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003523988-A 2003-08-12 JP claimed
EP-1263711-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES AstraZeneca AB (SE) 2002-12-11 EP claimed
WO-2001062704-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES ASTRAZENECA AB (SE) 2001-08-30 WO claimed
EP-1263711-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES AstraZeneca AB (SE) 2002-12-11 EP disclosed
WO-2001062704-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES ASTRAZENECA AB (SE) 2001-08-30 WO disclosed