SCHEMBL7606300

SCHEMBL7606300

Nc1ccc(-c2c(Cl)ccc(Sc3ccc(Cl)c(-c4ccc(N)cc4C(F)(F)F)c3Cl)c2Cl)c(C(F)(F)F)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.53
GLA P06280 1/20 0.53
POLB P06746 1/20 0.53
GAA P10253 1/20 0.53
ITGB2 P05107 2/20 0.40
ICAM1 P05362 2/20 0.40
ITGAL P20701 2/20 0.40
PDE7A Q13946 2/20 0.37
CYP3A4 P08684 1/20 0.34
IDO1 P14902 2/20 0.34
HTR3E A5X5Y0 1/20 0.34
HTR3B O95264 1/20 0.34
HTR3A P46098 1/20 0.34
HTR3D Q70Z44 1/20 0.34
HTR3C Q8WXA8 1/20 0.34
TRPV1 Q8NER1 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NOTUM Q6P988 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7610320 0.82 ITGB2 (0.50) TSHRPOLBGAAITGB2ICAM1
SCHEMBL7607008 0.81 ITGB2 (0.42) TSHRGLAPOLBGAAITGB2
SCHEMBL7610000 0.78 PDE7A (0.49) PDE7A
SCHEMBL30574189 0.76 TSHR (0.61) TSHRGLAPOLBGAACYP3A4
SCHEMBL203216 0.76 TSHR (0.61) TSHRGLAPOLBGAACYP3A4
SCHEMBL709679 0.74 GAA (0.59) TSHRGLAPOLBGAAITGB2
Hydrochloric Acid SCHEMBL9827180 0.74 TSHR (0.59) TSHRGLAPOLBGAAITGB2
Fluoride SCHEMBL10883445 0.74 TSHR (0.59) TSHRGLAPOLBGAACYP3A4
Hydrochloric Acid SCHEMBL4383138 0.74 TSHR (0.59) TSHRGLAPOLBGAAITGB2
Methane SCHEMBL27686801 0.72 TSHR (0.57) TSHRGLAPOLBGAACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165504-A2 INHIBITORS OF LFA-1 BINDING TO ICAMs AND USES THEREOF ICOS CORPORATION (US) 2002-01-02 EP disclosed
WO-2000059878-A2 INHIBITORS OF LFA-1 BINDING TO ICAMs AND USES THEREOF ICOS CORPORATION (US) 2000-10-12 WO disclosed