SCHEMBL7607008

SCHEMBL7607008

Nc1ccc(-c2c(Cl)ccc(Sc3ccc(Cl)c(-c4ccc(N)cc4F)c3Cl)c2Cl)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 2/20 0.42
ICAM1 P05362 2/20 0.42
ITGAL P20701 2/20 0.42
PDE7A Q13946 2/20 0.40
CYP3A4 P08684 3/20 0.37
TSHR P16473 2/20 0.37
KIT P10721 2/20 0.32
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
CYP2C19 P33261 1/20 0.31
KMT2A Q03164 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
ALDH1A1 P00352 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
GLA P06280 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7610320 0.85 ITGB2 (0.50) ITGB2ICAM1ITGALPDE7ACYP3A4
SCHEMBL7606300 0.81 TSHR (0.53) ITGB2ICAM1ITGALPDE7ACYP3A4
SCHEMBL7605576 0.76 PDE7A (0.48) PDE7AMAPTALDH1A1
SCHEMBL7610172 0.72 ITGB2 (0.50) ITGB2ICAM1ITGALPDE7ACYP3A4
SCHEMBL7606214 0.72 ITGB2 (0.50) ITGB2ICAM1ITGALPDE7ACYP3A4
Hydrochloric Acid SCHEMBL7605651 0.71 ITGB2 (0.53) ITGB2ICAM1ITGALPDE7ACYP3A4
SCHEMBL18860366 0.70 EPHB4 (0.39) CYP3A4TSHRKITKDM4EMAPT
SCHEMBL7610148 0.70 ITGB2 (0.47) ITGB2ICAM1ITGALPDE7ACYP3A4
SCHEMBL13385808 0.69 TSHR (0.41) CYP3A4TSHRKITKDM4EMEN1
SCHEMBL240923 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165504-A2 INHIBITORS OF LFA-1 BINDING TO ICAMs AND USES THEREOF ICOS CORPORATION (US) 2002-01-02 EP disclosed
WO-2000059878-A2 INHIBITORS OF LFA-1 BINDING TO ICAMs AND USES THEREOF ICOS CORPORATION (US) 2000-10-12 WO disclosed