SCHEMBL7606591

SCHEMBL7606591

COC(=O)Cc1ccccc1O.c1ccc2c(c1)C2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.50
EGFR P00533 3/20 0.43
TSHR P16473 3/20 0.42
KDM4E B2RXH2 2/20 0.42
MAPT P10636 1/20 0.41
ALDH1A1 P00352 4/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA7 P43166 1/20 0.40
CA14 Q9ULX7 1/20 0.40
NOTUM Q6P988 1/20 0.40
GAA P10253 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
NOX4 Q9NPH5 1/20 0.40
ATM Q13315 1/20 0.40
LMNA P02545 2/20 0.40
GFER P55789 1/20 0.40
CYP2D6 P10635 1/20 0.39
HIF1A Q16665 1/20 0.39
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL392976 0.90 AKR1B1 (0.61) AKR1B1EGFRTSHRKDM4EMAPT
SCHEMBL30311288 0.90 AKR1B1 (0.61) AKR1B1EGFRTSHRKDM4EMAPT
Methane SCHEMBL9292057 0.88 AKR1B1 (0.59) AKR1B1EGFRTSHRKDM4EMAPT
Phenol SCHEMBL2808100 0.83 AKR1B1 (0.58) AKR1B1EGFRTSHRKDM4EMAPT
SCHEMBL1554320 0.78 KDM4E (0.53) EGFRTSHRKDM4EMAPTALDH1A1
SCHEMBL21437933 0.77 PNMT (0.54) TSHRKDM4EMAPTALDH1A1NOTUM
SCHEMBL9755818 0.76 NOTUM (0.51) TSHRKDM4EMAPTALDH1A1CA12
SCHEMBL607310 0.76 NPC1 (0.52) AKR1B1TSHRKDM4EMAPTALDH1A1
SCHEMBL29852765 0.76 NPC1 (0.52) AKR1B1TSHRKDM4EMAPTALDH1A1
SCHEMBL25285645 0.76 IAPP (0.51) AKR1B1EGFRKDM4EMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6395919-B1 Calcilytic compounds SMITHKLINE BEECHAM CORPORATION 2002-05-28 US disclosed
EP-1070048-A4 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2001-11-07 EP disclosed
EP-1070048-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2001-01-24 EP disclosed
WO-1999051569-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1999-10-14 WO disclosed