SCHEMBL7607538

SCHEMBL7607538

COc1ccc2c(c1)OCCC(CN(C)C)=C2c1cccc(O)c1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 17/20 0.47
ESR2 Q92731 17/20 0.47
CYP19A1 P11511 1/20 0.42
MAOB P27338 1/20 0.37
GRM5 P41594 1/20 0.37
HSD17B1 P14061 1/20 0.37
HSD17B2 P37059 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8016453 0.99 ESR1 (0.46) ESR1ESR2CYP19A1MAOBGRM5
SCHEMBL7604532 0.89 MAOA (0.45) ESR1ESR2MAOB
Hydrochloric Acid SCHEMBL8018596 0.88 MAOA (0.44) ESR1ESR2MAOB
SCHEMBL7611354 0.87 MAOB (0.53) ESR1ESR2MAOBGRM5
Hydrochloric Acid SCHEMBL8022844 0.86 MAOB (0.53) ESR1ESR2MAOBGRM5
SCHEMBL7605971 0.85 ESR1 (0.49) ESR1ESR2
SCHEMBL7605210 0.84 ESR1 (0.44) ESR1ESR2
Hydrochloric Acid SCHEMBL8016456 0.84 ESR1 (0.49) ESR1ESR2
Hydrochloric Acid SCHEMBL8016570 0.83 ESR1 (0.43) ESR1ESR2
SCHEMBL7611830 0.81 OPRD1 (0.35) ESR1ESR2MAOBHSD17B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0922703-B1 Substituted heterocyclic benzocycloalkenes and their use as analgesically active compounds GRUENENTHAL GMBH (DE) 2002-12-04 EP disclosed
EP-0917545-B1 PRESSURE SENSITIVE MATERIALS WITH SMALL AMOUNTS OF STYRENE BASF AG (DE) 2002-04-10 EP disclosed
EP-0917546-B1 PRESSURE SENSITIVE MATERIALS BASED ON MULTISTEP CONSTITUTED OF POLYMERIZATES BASF AG (DE) 2001-06-06 EP disclosed
EP-0922703-A1 Substituted heterocyclic benzocycloalkenes and their use as analgesically active compounds Grünenthal GmbH (DE) 1999-06-16 EP disclosed