SCHEMBL7607691

SCHEMBL7607691

COc1nc(N)nc(OC)c1Cl

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCNA2 P20248 1/20 0.47
CDK2 P24941 1/20 0.47
CCNA1 P78396 1/20 0.47
CYP1A2 P05177 1/20 0.42
HSP90AA1 P07900 9/20 0.35
HSP90AB1 P08238 8/20 0.35
MAPT P10636 2/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PDCD1LG2 Q9BQ51 4/20 0.33
CD274 Q9NZQ7 4/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CHRM4 P08173 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8008714 0.88 CYP1A2 (0.52) CCNA2CDK2CCNA1CYP1A2HSP90AA1
SCHEMBL28221808 0.86 CCNA2 (0.41) CCNA2CDK2CCNA1CYP1A2HSP90AA1
SCHEMBL16828162 0.78 CCNA2 (0.50) CCNA2CDK2CCNA1
SCHEMBL9432184 0.78 CYP1A2 (0.61) CYP1A2MAPTGAASMN1; SMN2PDCD1LG2
SCHEMBL11059135 0.77 CCNA2 (0.46) CCNA2CDK2CCNA1CYP1A2HSP90AA1
SCHEMBL30559673 0.77 CCNA2 (0.46) CCNA2CDK2CCNA1CYP1A2HSP90AA1
SCHEMBL26977474 0.77 CCNA2 (0.46) CCNA2CDK2CCNA1CYP1A2HSP90AA1
SCHEMBL10617813 0.76 CCNA2 (0.48) CCNA2CDK2CCNA1HSP90AA1HSP90AB1
SCHEMBL30721418 0.76 CCNA2 (0.48) CCNA2CDK2CCNA1HSP90AA1HSP90AB1
Hydrochloric Acid SCHEMBL16828222 0.76 CCNA2 (0.48) CCNA2CDK2CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6087500-A Methods for producing pyrimidine compounds NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2000-07-11 US claimed
EP-0902019-A1 PROCESSES FOR THE PREPARATION OF PYRIMIDINE COMPOUND NISSAN CHEMICAL INDUSTRIES, LIMITED (JP) 1999-03-17 EP claimed
EP-4744661-A2 NOVEL PYRIMIDIN-2-YL SULFONAMIDE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2026-05-20 EP disclosed
EP-4298092-B1 NOVEL PYRIMIDIN-2-YL SULFONAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2025-11-26 EP disclosed
US-20240025883-A1 PYRIMIDIN-2-YL SULFONAMIDE DERIVATIVES HOFFMANN-LA ROCHE INC. (US) 2024-01-25 US disclosed
US-20240025883-A1 PYRIMIDIN-2-YL SULFONAMIDE DERIVATIVES HOFFMANN-LA ROCHE INC. (US) 2024-01-25 US disclosed
US-20240025883-A1 PYRIMIDIN-2-YL SULFONAMIDE DERIVATIVES HOFFMANN-LA ROCHE INC. (US) 2024-01-25 US disclosed
CN-116829550-A Pyrimidine-2-ylsulfonamide derivatives 豪夫迈·罗氏有限公司 2023-09-29 CN disclosed
EP-0902019-A4 PROCESSES FOR THE PREPARATION OF PYRIMIDINE COMPOUND NISSAN CHEMICAL IND LTD (JP) 2002-03-27 EP disclosed
US-6087500-A Methods for producing pyrimidine compounds NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2000-07-11 US disclosed
US-6087500-A Methods for producing pyrimidine compounds NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2000-07-11 US disclosed
EP-0902019-A1 PROCESSES FOR THE PREPARATION OF PYRIMIDINE COMPOUND NISSAN CHEMICAL INDUSTRIES, LIMITED (JP) 1999-03-17 EP disclosed
EP-0902019-A1 PROCESSES FOR THE PREPARATION OF PYRIMIDINE COMPOUND NISSAN CHEMICAL INDUSTRIES, LIMITED (JP) 1999-03-17 EP disclosed
WO-1997043265-A1 PROCESSES FOR THE PREPARATION OF PYRIMIDINE COMPOUND NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1997-11-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240025883-A1 PYRIMIDIN-2-YL SULFONAMIDE DERIVATIVES GPR17, GPR27, GPR119 CCNA2 2260/4885CDK2 1005/4885CCNA1 2045/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.