SCHEMBL7608430

SCHEMBL7608430

Cc1cccc(CC(=O)N2CCN(CCCCC3(OC(=O)NCC(F)(F)F)c4ccccc4-c4ccccc43)CC2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.43
POLB P06746 1/20 0.43
RECQL P46063 1/20 0.40
CHRM2 P08172 1/20 0.39
ADRA2A P08913 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
CHRM1 P11229 1/20 0.39
DRD1 P21728 1/20 0.39
TBXA2R P21731 1/20 0.39
PTGS1 P23219 1/20 0.39
SLC6A2 P23975 1/20 0.39
ADRA1A P35348 1/20 0.39
OPRM1 P35372 1/20 0.39
DRD3 P35462 1/20 0.39
MTTP P55157 1/20 0.39
SLC6A3 Q01959 1/20 0.39
KCNH2 Q12809 1/20 0.39
MTR Q99707 1/20 0.39
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7634068 0.91 SIGMAR1 (0.42) SIGMAR1CHRM2ADRA2AADORA3CHRM1
SCHEMBL6675771 0.91 SIGMAR1 (0.45) SIGMAR1CHRM2ADRA2AADORA3CHRM1
SCHEMBL7610087 0.90 ATM (0.44) SIGMAR1CHRM2ADRA2AADORA3CHRM1
SCHEMBL7605238 0.90 MEN1 (0.48) SIGMAR1CHRM2ADRA2AADORA3CHRM1
SCHEMBL7611938 0.88 SIGMAR1 (0.46) SIGMAR1ALDH1A1KDM4E
SCHEMBL7637370 0.88 SIGMAR1 (0.42) SIGMAR1CHRM2ADRA2AADORA3CHRM1
SCHEMBL7638227 0.87 SIGMAR1 (0.44) SIGMAR1CHRM2ADRA2AADORA3CHRM1
SCHEMBL7049298 0.87 MTTP (0.51) POLBCHRM2ADRA2AADORA3CHRM1
SCHEMBL7611306 0.87 ADRA1A (0.42) SIGMAR1POLBCHRM2ADRA2AADORA3
SCHEMBL6678861 0.86 MTTP (0.50) SIGMAR1CHRM2ADRA2AADORA3CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1259492-A1 SUBSTITUTED PIPERAZINE DERIVATIVES AS MTP INHIBITORS Boehringer Ingelheim Pharma KG (DE) 2002-11-27 EP disclosed
WO-2001047899-A1 SUBSTITUTED PIPERAZINE DERIVATIVES AS MTP INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-07-05 WO disclosed