SCHEMBL7608863

SCHEMBL7608863

O=C1[CH]c2cccnc2C=C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
S100A4 P26447 1/20 0.35
CDC25B P30305 1/20 0.35
BLM P54132 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
TDP2 O95551 1/20 0.34
NSD2 O96028 1/20 0.34
ABL1 P00519 1/20 0.34
PLCG1 P19174 1/20 0.34
CES1 P23141 1/20 0.34
PAX8 Q06710 1/20 0.34
RIN1 Q13671 1/20 0.34
MEN1 O00255 1/20 0.34
THRB P10828 1/20 0.34
KMT2A Q03164 1/20 0.34
GAA P10253 1/20 0.34
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3261185 0.82
SCHEMBL2074744 0.74
SCHEMBL1648797 0.71 CA12 (0.42) CA12CA1CA2CA9S100A4
SCHEMBL1648800 0.71 CA12 (0.42) CA12CA1CA2CA9S100A4
SCHEMBL27847095 0.70 CA12 (0.41) CA12CA1CA2CA9S100A4
Iodide SCHEMBL3908355 0.70 CA12 (0.41) CA12CA1CA2CA9S100A4
Iodide SCHEMBL3908349 0.70 CA12 (0.41) CA12CA1CA2CA9S100A4
SCHEMBL23330240 0.68 CA12 (0.44) CA12CA1CA2CA9S100A4
SCHEMBL15800569 0.68 CA12 (0.40) CA12CA1CA2CA9S100A4
SCHEMBL1927673 0.67 MAPT (0.46) CDC25BBLMTDP1CES1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1254164-A2 SELECTIVE N-ACYLATION OF A82846 GLYCOPEPTIDE ANALOGS ELI LILLY AND COMPANY (US) 2002-11-06 EP disclosed
WO-2001058933-A2 SELECTIVE N-ACYLATION OF A82846 GLYCOPEPTIDE ANALOGS ELI LILLY AND COMPANY (US) 2001-08-16 WO disclosed