SCHEMBL7610982

SCHEMBL7610982

CCN(C)C(=O)OC1(CCCCBr)c2ccccc2-c2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 9/20 0.40
TSPO P30536 2/20 0.35
SCN1A P35498 2/20 0.33
SCN2A Q99250 2/20 0.33
SCN3A Q9NY46 2/20 0.33
APEX1 P27695 1/20 0.33
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7595167 0.80 APEX1 (0.41) PDK2APEX1
SCHEMBL7612764 0.79 MAPT (0.38) PDK2APEX1
SCHEMBL7595150 0.79 APEX1 (0.37) APEX1
SCHEMBL7600206 0.79 PDK2 (0.39) PDK2
SCHEMBL7046510 0.78 PDK2 (0.43) PDK2APEX1
SCHEMBL7595652 0.77 PDK2 (0.41) PDK2
SCHEMBL7613371 0.75 SIGMAR1 (0.47)
SCHEMBL7597301 0.73 KMT2A (0.39) APEX1
SCHEMBL7599983 0.73 PDK2 (0.37) PDK2
SCHEMBL7599929 0.72 TP53 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1259492-A1 SUBSTITUTED PIPERAZINE DERIVATIVES AS MTP INHIBITORS Boehringer Ingelheim Pharma KG (DE) 2002-11-27 EP disclosed
WO-2001047899-A1 SUBSTITUTED PIPERAZINE DERIVATIVES AS MTP INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-07-05 WO disclosed