SCHEMBL761446

SCHEMBL761446

CC(=O)NCCc1cccc2ccccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 18/20 0.73
MTNR1B P49286 14/20 0.73
NQO2 P16083 5/20 0.66
HTR2C P28335 1/20 0.66
HTR2B P41595 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29941181 1.00 MTNR1A (0.73) MTNR1AMTNR1BNQO2HTR2CHTR2B
SCHEMBL1846496 0.86 MTNR1A (0.67) MTNR1AMTNR1BNQO2HTR2CHTR2B
SCHEMBL1567114 0.85 MTNR1A (0.73) MTNR1AMTNR1BNQO2
SCHEMBL7016328 0.84 MTNR1A (1.00) MTNR1AMTNR1BNQO2HTR2CHTR2B
SCHEMBL2608948 0.84 MTNR1A (0.68) MTNR1AMTNR1BNQO2
SCHEMBL8065745 0.84 MTNR1A (0.68) MTNR1ANQO2
SCHEMBL5511489 0.83 MTNR1A (1.00) MTNR1AMTNR1BNQO2
SCHEMBL4043404 0.83 MTNR1A (1.00) MTNR1AMTNR1BNQO2HTR2CHTR2B
SCHEMBL1688124 0.83 MTNR1A (0.77) MTNR1AMTNR1BNQO2HTR2CHTR2B
SCHEMBL30449793 0.83 MTNR1A (1.00) MTNR1AMTNR1BNQO2HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104178546-B The method of optical voidness S-1-naphthalene ethylamine is prepared in a kind of fractionation CHEN YONGJUN (CN) 2017-01-04 CN claimed
CN-104164470-B The method of optical voidness R-1-naphthalene ethylamine is prepared in a kind of fractionation 六安佳诺生化科技有限公司 2016-12-21 CN claimed
CN-104178547-B The method of optical voidness S-1-naphthalene ethylamine is prepared in a kind of fractionation 陈永军 2016-12-07 CN claimed
CN-104151171-B The method of optical voidness R-1-naphthalene ethylamine is prepared in a kind of fractionation 六安佳诺生化科技有限公司 2016-07-27 CN claimed
CN-104178546-A Method for preparing optically-pure S-1-naphthylethylamine through resolution CHEN YONGJUN 2014-12-03 CN claimed
CN-104178547-A Method for preparing optically-pure S-1-naphthylethylamine through resolution CHEN YONGJUN 2014-12-03 CN claimed
CN-104164470-A Method for preparing optically pure R-1-naphthylethylamine by resolution CHEN YONGJUN 2014-11-26 CN claimed
CN-104151171-A Method for preparing optically pure R-1-naphthylethylamine by splitting CHEN YONGJUN 2014-11-19 CN claimed
EP-3551639-A1 NOVEL CHIRAL DIHYDROBENZOAZAPHOSPHOLE LIGANDS AND SYNTHESIS THEREOF Boehringer Ingelheim International GmbH (DE) 2019-10-16 EP disclosed
WO-2018106621-A1 NOVEL CHIRAL DIHYDROBENZOAZAPHOSPHOLE LIGANDS AND SYNTHESIS THEREOF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-06-14 WO disclosed
CN-104178546-B The method of optical voidness S-1-naphthalene ethylamine is prepared in a kind of fractionation CHEN YONGJUN (CN) 2017-01-04 CN disclosed
CN-104178546-B The method of optical voidness S-1-naphthalene ethylamine is prepared in a kind of fractionation CHEN YONGJUN (CN) 2017-01-04 CN disclosed
CN-104164470-B The method of optical voidness R-1-naphthalene ethylamine is prepared in a kind of fractionation 六安佳诺生化科技有限公司 2016-12-21 CN disclosed
CN-104178547-B The method of optical voidness S-1-naphthalene ethylamine is prepared in a kind of fractionation 陈永军 2016-12-07 CN disclosed
WO-2001007409-A1 CARBAZOLE DERIVATIVES AND THEIR USE AS NEUROPEPTIDE Y5 RECEPTOR LIGANDS ASTRAZENECA UK LIMITED (GB) 2001-02-01 WO disclosed
WO-1999058496-A1 NOVEL SUBSTITUTED CYCLIC COMPOUNDS, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ADIR ET COMPAGNIE (FR) 1999-11-18 WO disclosed
US-5616614-A USEFUL IN TREATMENT OF DISORDERS LINKED TO ABNORMAL MELATONIN ACTIVITY ADIR ET COMPAGNIE (FR) 1997-04-01 US disclosed
EP-0562956-B1 Naphtylalkylamines, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1995-09-27 EP disclosed
US-5420158-A Melatonin activity ADIR ET COMPAGNIE (FR) 1995-05-30 US disclosed
EP-0562956-A1 Naphtylalkylamines, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1993-09-29 EP disclosed