SCHEMBL7615262

SCHEMBL7615262

C=CCN1CCC(Br)C1=O

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.35
ALDH1A1 P00352 1/20 0.33
ACE P12821 1/20 0.32
MAPT P10636 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
PIK3CD O00329 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC7 Q8WUI4 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC10 Q969S8 1/20 0.31
HDAC11 Q96DB2 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HDAC9 Q9UKV0 1/20 0.31
HDAC5 Q9UQL6 1/20 0.31
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7615273 1.00 CYP3A4 (0.35) CYP3A4ALDH1A1ACEMAPTL3MBTL1
SCHEMBL7615268 1.00 CYP3A4 (0.35) CYP3A4ALDH1A1ACEMAPTL3MBTL1
SCHEMBL26361631 0.79 FAAH (0.39) CYP3A4ALDH1A1ACEMAPTL3MBTL1
SCHEMBL9000514 0.78 CYP3A4 (0.37) CYP3A4ALDH1A1MAPTL3MBTL1PIK3CD
SCHEMBL4594212 0.77 PIK3CD (0.55) CYP3A4ALDH1A1MAPTL3MBTL1PIK3CD
SCHEMBL1682219 0.77 CYP3A4 (0.44) CYP3A4ALDH1A1MAPTL3MBTL1PIK3CD
SCHEMBL1551140 0.77 CYP3A4 (0.35) CYP3A4ALDH1A1ACEMAPTL3MBTL1
SCHEMBL7510369 0.76 FPR2 (0.35) ACEL3MBTL1PIK3CDNPSR1
SCHEMBL7619079 0.76 FPR2 (0.35) ACEL3MBTL1PIK3CDNPSR1
SCHEMBL7619075 0.76 FPR2 (0.35) ACEL3MBTL1PIK3CDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620225-B1 Cephalosporin derivatives BASILEA PHARMACEUTICA AG (CH) 2002-11-13 EP disclosed
US-5523400-A 3-(PYRROLIDIN-3-YLIDENE=CH-),7-((2-AMINOTHIAZOL-4-YL)HYDROX -IMINOACETYLAMINO-)-3-CEPHEM DERIVATIVES; BROAD SPECTRUM ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1996-06-04 US disclosed
EP-0620225-A1 Cephalosporin derivatives F. HOFFMANN-LA ROCHE AG (CH) 1994-10-19 EP disclosed