Piperidine

Piperidine

SCHEMBL7619489

C1CCNCC1.O=Cc1ccccc1C(=O)O

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 4/20 0.43
ALOX15 P16050 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
STS P08842 4/20 0.39
TDP1 Q9NUW8 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
LMNA P02545 2/20 0.39
THRB P10828 1/20 0.39
BLM P54132 1/20 0.39
ABCC1 P33527 1/20 0.38
GRIK1 P39086 1/20 0.38
GRIA1 P42261 1/20 0.38
GRIA2 P42262 1/20 0.38
GRIA3 P42263 1/20 0.38
GRIA4 P48058 1/20 0.38
GRIK2 Q13002 1/20 0.38
GRIK3 Q13003 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyrrolidine SCHEMBL15054617 0.98 ALDH1A1 (0.44) ALDH1A1KDM4EALOX15CYP1A2CYP2C9
Piperidine SCHEMBL7621076 0.88 MEN1 (0.40) ALDH1A1KDM4ETDP1MEN1KMT2A
Phthalic Acid SCHEMBL5875074 0.84 ALDH1A1 (0.61) ALDH1A1KDM4EALOX15TDP1ABCC1
Phthalic Acid SCHEMBL5875064 0.84 ALDH1A1 (0.61) ALDH1A1KDM4EALOX15TDP1ABCC1
SCHEMBL78873 0.84 ALDH1A1 (0.59) ALDH1A1KDM4EALOX15CYP1A2CYP2C9
SCHEMBL29556927 0.84 ALDH1A1 (0.59) ALDH1A1KDM4EALOX15CYP1A2CYP2C9
Benzene SCHEMBL28103329 0.84 ALDH1A1 (0.59) ALDH1A1KDM4EALOX15CYP1A2CYP2C9
SCHEMBL20448823 0.84 ALDH1A1 (0.59) ALDH1A1KDM4EALOX15CYP1A2CYP2C9
Hydrochloric Acid SCHEMBL7536438 0.82 ALDH1A1 (0.56) ALDH1A1KDM4EALOX15CYP1A2CYP2C9
Phthalic Acid SCHEMBL29243281 0.82 ALDH1A1 (0.64) ALDH1A1KDM4EALOX15CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0635004-B1 4-DIPHENYLMETHYL PIPERIDINE DERIVATIVES AND PROCESS FOR THEIR PREPARATION MERRELL PHARMA INC (US) 2002-07-17 EP claimed
US-5675009-A Process for piperidine derivatives MERRELL PHARMACEUTICALS INC. (US) 1997-10-07 US claimed
US-5644061-A Process for piperidine derivatives MERRELL PHARMACEUTICALS INC. (US) 1997-07-01 US claimed
EP-0635004-A1 4-DIPHENYLMETHYL PIPERIDINE DERIVATIVES AND PROCESS FOR THEIR PREPARATION MERRELL PHARMACEUTICALS INC. (US) 1995-01-25 EP claimed
WO-1993021156-A1 4-DIPHENYLMETHYL PIPERIDINE DERIVATIVES AND PROCESS FOR THEIR PREPARATION MERRELL DOW PHARMACEUTICALS INC. (US) 1993-10-28 WO claimed
EP-0635004-B1 4-DIPHENYLMETHYL PIPERIDINE DERIVATIVES AND PROCESS FOR THEIR PREPARATION MERRELL PHARMA INC (US) 2002-07-17 EP disclosed
US-5675009-A Process for piperidine derivatives MERRELL PHARMACEUTICALS INC. (US) 1997-10-07 US disclosed
US-5663353-A Process for piperidine derivatives MERRELL PHARMACEUTICALS INC. (US) 1997-09-02 US disclosed
US-5654433-A Process for piperidine derivatives MERRELL PHARMACEUTICALS INC. (US) 1997-08-05 US disclosed
US-5652370-A Process for piperidine derivatives MERRELL PHARMACEUTICALS INC. (US) 1997-07-29 US disclosed
US-5650516-A Process for piperidine derivatives MERRELL PHARMACEUTICALS INC. (US) 1997-07-22 US disclosed
US-5644061-A Process for piperidine derivatives MERRELL PHARMACEUTICALS INC. (US) 1997-07-01 US disclosed
US-5631375-A Process for piperidine derivatives MERRELL PHARMACEUTICALS, INC. (US) 1997-05-20 US disclosed
US-5618940-A Process for piperidine derivatives MERRELL PHARMACEUTICALS INC. (US) 1997-04-08 US disclosed
EP-0635004-A1 4-DIPHENYLMETHYL PIPERIDINE DERIVATIVES AND PROCESS FOR THEIR PREPARATION MERRELL PHARMACEUTICALS INC. (US) 1995-01-25 EP disclosed
WO-1993021156-A1 4-DIPHENYLMETHYL PIPERIDINE DERIVATIVES AND PROCESS FOR THEIR PREPARATION MERRELL DOW PHARMACEUTICALS INC. (US) 1993-10-28 WO disclosed