SCHEMBL7624883

SCHEMBL7624883

COc1ccc2c(c1)CCC(Br)=C2c1ccc(O)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 7/20 0.60
ESR2 Q92731 3/20 0.58
MIF P14174 4/20 0.54
CYP26A1 O43174 3/20 0.54
CYP24A1 Q07973 1/20 0.45
KDM4E B2RXH2 2/20 0.44
GLA P06280 2/20 0.44
CYP27A1 Q02318 1/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
RAB9A P51151 1/20 0.43
ATM Q13315 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ALKBH3 Q96Q83 1/20 0.43
IDH1 O75874 1/20 0.42
EBP Q15125 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
ABL1 P00519 1/20 0.41
ABCB1 P08183 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20165138 0.89 ESR1 (0.54) ESR1ESR2MIFCYP26A1KDM4E
SCHEMBL29756936 0.89 ESR1 (0.54) ESR1ESR2MIFCYP26A1KDM4E
SCHEMBL29632065 0.85 ESR1 (0.46) ESR1ESR2MIFCYP26A1CYP24A1
SCHEMBL20211917 0.85 ESR1 (0.46) ESR1ESR2MIFCYP26A1CYP24A1
SCHEMBL7623247 0.83 ESR1 (0.75) ESR1ESR2MIFCYP26A1EBP
SCHEMBL18850173 0.83 ESR1 (0.52) ESR1ESR2MIFGAAMAPT
SCHEMBL115122 0.83 EBP (0.47) ESR1ESR2MIFCYP26A1CYP24A1
SCHEMBL7633352 0.83 MIF (0.48) ESR1ESR2MIFCYP26A1CYP27A1
SCHEMBL23297257 0.81 EBP (0.51) ESR1MIFCYP26A1CYP27A1MAPT
SCHEMBL18845516 0.81 ESR1 (0.51) ESR1ESR2MIFALKBH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0955286-B1 Dihydro- or tetrahydronaphthalene derivatives having (anti-)estrogen activity AVENTIS PHARMA SA (FR) 2002-08-07 EP disclosed
US-6005003-A OSTEOPOROSIS TREATMENT HOECHST MARION ROUSSEL (FR) 1999-12-21 US disclosed
EP-0955286-A1 Dihydro- or tetrahydronaphthalene derivatives having (anti-)estrogen activity HOECHST MARION ROUSSEL (FR) 1999-11-10 EP disclosed