SCHEMBL7625943

SCHEMBL7625943

O=C1C(Cc2ccccc2)NC(c2ccccc2)=CN1O

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.47
POLB P06746 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C19 P33261 1/20 0.47
PLA2G10 O15496 2/20 0.46
PLA2G5 P39877 2/20 0.46
ALDH1A1 P00352 1/20 0.42
HDAC1 Q13547 3/20 0.41
HDAC6 Q9UBN7 3/20 0.41
HDAC8 Q9BY41 2/20 0.41
CES2 O00748 1/20 0.40
ALOX15 P16050 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7616025 0.97 GAA (0.45) GAAPOLBCYP1A2CYP3A4CYP2C19
SCHEMBL7622610 0.94 GAA (0.43) GAAPOLBCYP1A2CYP3A4CYP2C19
SCHEMBL7615634 0.94 GAA (0.43) GAAPOLBCYP1A2CYP3A4CYP2C19
SCHEMBL7625933 0.92 GAA (0.50) GAAPOLBCYP1A2CYP3A4CYP2C19
SCHEMBL7619044 0.91 NPSR1 (0.49) GAAPOLBCYP1A2CYP3A4CYP2C19
SCHEMBL7617539 0.91 ALDH1A1 (0.52) GAAPOLBCYP1A2CYP3A4CYP2C19
SCHEMBL7623410 0.91 CES2 (0.45) GAAPOLBCYP1A2CYP3A4CYP2C19
SCHEMBL7616794 0.88 NPSR1 (0.45) GAAPOLBCYP1A2CYP3A4CYP2C19
SCHEMBL7591446 0.88 CES2 (0.44) GAAPOLBCYP1A2CYP3A4CYP2C19
SCHEMBL7616578 0.88 ALDH1A1 (0.47) GAAPOLBCYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436933-B1 1-HYDROXY-3-(2-METHYLPROPYL)-5,6-DIPHENYLHYDROPYRAZIN-2-ONE STRUCTURAL BIOINFORMATICS INC. 2002-08-20 US claimed
US-6436933-B1 1-HYDROXY-3-(2-METHYLPROPYL)-5,6-DIPHENYLHYDROPYRAZIN-2-ONE STRUCTURAL BIOINFORMATICS INC. 2002-08-20 US disclosed