Iodide

Iodide

SCHEMBL7628545

CCOc1ccc(-c2ccc3c(c2)C=C(C(=O)Nc2ccc(CC4OCCC(C)(N)C4C)cc2)CCO3)cc1.I

nearest known ligand 0.61

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNG

The experimentally established mechanism targets of Iodide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 19/20 0.61
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL5247643 0.92 CCR5 (0.53) CCR5
Iodide SCHEMBL7624169 0.88 CCR5 (0.60) CCR5
Iodide SCHEMBL7925879 0.86 CCR5 (0.51) CCR5
SCHEMBL5204397 0.81 CCR5 (0.72) CCR5NPC1RAB9A
SCHEMBL5205911 0.81 CCR5 (0.71) CCR5NPC1RAB9A
Iodide SCHEMBL7678820 0.79 CCR5 (0.59) CCR5
Iodide SCHEMBL7619257 0.76 CCR5 (0.62) CCR5
SCHEMBL5208604 0.76 CCR5 (0.63) CCR5
Iodide SCHEMBL7681114 0.76 CCR5 (0.63) CCR5
SCHEMBL3034760 0.76 CCR5 (0.73) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6413947-B1 Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-02 US disclosed
US-6376536-B1 VIRICIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-04-23 US disclosed
US-6268354-B1 Pharmaceutical composition for antagonizing CCR5 comprising anilide derivative TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-07-31 US disclosed
EP-1104416-A2 QUATERNARY AMMONIUM SALTS AND THEIR USE AS ANTI-HIV AGENTS Takeda Chemical Industries, Ltd. (JP) 2001-06-06 EP disclosed
US-6166006-A Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-12-26 US disclosed
US-6096780-A ANTIVIRAL COMPOUND USEFUL FOR TREATING HIV VIRUSES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-08-01 US disclosed
WO-2000010965-A2 QUATERNARY AMMONIUM SALTS AND THEIR USE AS ANTI-HIV AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-03-02 WO disclosed