Iodide

Iodide

SCHEMBL7681114

CC1C(Cc2ccc(NC(=O)C3=Cc4cc(-c5ccc(N6CCCCC6)cc5)ccc4CCC3)cc2)OCCC1(C)N.I

nearest known ligand 0.63

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNG

The experimentally established mechanism targets of Iodide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 18/20 0.63
CCR2 P41597 3/20 0.49
CXCR3 P49682 3/20 0.49
CCR7 P32248 2/20 0.49
CXCR5 P32302 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL7619257 0.99 CCR5 (0.62) CCR5CCR2CXCR3CCR7CXCR5
Iodide SCHEMBL7925879 0.89 CCR5 (0.51) CCR5
Iodide SCHEMBL5247643 0.79 CCR5 (0.53) CCR5
SCHEMBL5208811 0.77 CCR2 (0.81) CCR5CCR2CXCR3CCR7CXCR5
Iodide SCHEMBL7681118 0.77 CCR5 (1.00) CCR5CCR2CXCR3CCR7CXCR5
Iodide SCHEMBL7624169 0.76 CCR5 (0.60) CCR5
SCHEMBL5240554 0.76 CCR2 (0.82) CCR5CCR2CXCR3CCR7CXCR5
Iodide SCHEMBL7628545 0.76 CCR5 (0.61) CCR5
Iodide SCHEMBL5204391 0.76 CCR5 (1.00) CCR5CCR2CXCR3CCR7CXCR5
SCHEMBL5208454 0.71 CCR5 (0.70) CCR5CCR2CXCR3CCR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6413947-B1 Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-02 US disclosed
US-6268354-B1 Pharmaceutical composition for antagonizing CCR5 comprising anilide derivative TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-07-31 US disclosed
US-6166006-A Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-12-26 US disclosed
EP-1040103-A1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-10-04 EP disclosed
WO-1999032468-A1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-07-01 WO disclosed