SCHEMBL763040

SCHEMBL763040

CC(=O)NCCn1c([C@@H]2CCCN(C(=O)C[C@H](N)Cc3ccc(-c4ccc5c(c4)NC(=O)CO5)cc3)C2)nc2ccccc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
RXFP1 Q9HBX9 1/20 0.38
HRH1 P35367 5/20 0.38
CYP2D6 P10635 4/20 0.38
PIK3CA P42336 1/20 0.38
DGAT2 Q96PD7 1/20 0.37
PARP1 P09874 1/20 0.37
CTSC P53634 1/20 0.36
CPT1A P50416 3/20 0.36
CPT2 P23786 2/20 0.36
CPT1B Q92523 2/20 0.36
MMP8 P22894 2/20 0.36
MMP13 P45452 2/20 0.36
KCNH2 Q12809 3/20 0.35
CHRM1 P11229 2/20 0.35
CXCR3 P49682 1/20 0.35
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740643 0.90 HRH1 (0.39) HRH1CYP2D6CTSCKCNH2CHRM1
SCHEMBL740644 0.90 HRH1 (0.39) HRH1CYP2D6CTSCKCNH2CHRM1
SCHEMBL742247 0.89 MAPT (0.39) MAPTALDH1A1LMNARXFP1HRH1
SCHEMBL742248 0.89 MAPT (0.39) MAPTALDH1A1LMNARXFP1HRH1
SCHEMBL741495 0.89 HRH1 (0.39) HRH1CYP2D6KCNH2CHRM1
SCHEMBL741496 0.89 HRH1 (0.39) HRH1CYP2D6KCNH2CHRM1
SCHEMBL740858 0.88 HRH1 (0.41) ALDH1A1LMNAHRH1CYP2D6KCNH2
SCHEMBL740859 0.88 HRH1 (0.41) ALDH1A1LMNAHRH1CYP2D6KCNH2
SCHEMBL739243 0.86 HRH1 (0.41) HRH1CYP2D6KCNH2CHRM1
SCHEMBL739242 0.86 HRH1 (0.41) HRH1CYP2D6KCNH2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed