SCHEMBL7633288

SCHEMBL7633288

NCC(CC(=O)O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.68

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GABBR2 O75899 5/20 0.68
GABBR1 Q9UBS5 5/20 0.68
LMNA P02545 2/20 0.68
CYP2C9 P11712 2/20 0.68
CYP3A4 P08684 1/20 0.68
ADORA3 P0DMS8 1/20 0.68
NFKB1 P19838 1/20 0.68
DRD3 P35462 1/20 0.68
BLM P54132 1/20 0.68
CYP1A2 P05177 1/20 0.68
CYP2D6 P10635 1/20 0.68
CYP2C19 P33261 1/20 0.68
MEN1 O00255 1/20 0.68
THRB P10828 1/20 0.68
TSHR P16473 1/20 0.68
KMT2A Q03164 1/20 0.68
GAA P10253 1/20 0.54
PRKCZ Q05513 2/20 0.50
FFAR1 O14842 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL560490 0.98 GABBR2 (0.66) GABBR2GABBR1LMNACYP2C9CYP3A4
Trifluoroacetic Acid SCHEMBL8903793 0.91 GABBR2 (0.57) GABBR2GABBR1LMNACYP2C9CYP3A4
SCHEMBL1532918 0.90 PRKCZ (0.54) GABBR2GABBR1LMNACYP2C9CYP3A4
SCHEMBL560574 0.87 GABBR2 (0.64) GABBR2GABBR1LMNACYP2C9CYP3A4
Hydrochloric Acid SCHEMBL560861 0.87 GABBR2 (0.56) GABBR2GABBR1LMNACYP2C9CYP3A4
SCHEMBL26231951 0.86 GABBR2 (0.62) GABBR2GABBR1LMNACYP2C9CYP3A4
SCHEMBL559899 0.86 GABBR2 (0.62) GABBR2GABBR1LMNACYP2C9CYP3A4
Hydrochloric Acid SCHEMBL560273 0.84 GABBR2 (0.60) GABBR2GABBR1LMNACYP2C9CYP3A4
SCHEMBL560445 0.84 GABBR2 (0.52) GABBR2GABBR1LMNACYP2C9CYP3A4
Hydrochloric Acid SCHEMBL559973 0.83 GABBR2 (0.51) GABBR2GABBR1LMNACYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6433174-B1 Process for producing novel naphthyridine derivatives NIPPON KAYAKU KABUSHIKI KAISHA (JP) 2002-08-13 US disclosed
EP-1142892-A1 PROCESSES FOR THE PREPARATION OF NOVEL NAPHTHYRIDINE DERIVATIVES Nippon Kayaku Kabushiki Kaisha (JP) 2001-10-10 EP disclosed
US-5686609-A Aromatic amine compounds, Their method of preparation and pharmaceutical compositions in which they are present SANOFI (FR) 1997-11-11 US disclosed
US-5618938-A Process for preparing stereo isomers of neurokinin receptor antagonists SANOFI (FR) 1997-04-08 US disclosed
US-5317020-A Neurokinin receiver antagonist as antiinflammatory agents SANOFI (FR) 1994-05-31 US disclosed