SCHEMBL763378

SCHEMBL763378

Cc1nc2ccccc2n1C1CCCNC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.53
JAK1 P23458 1/20 0.53
HDAC1 Q13547 3/20 0.51
HDAC8 Q9BY41 3/20 0.51
HDAC6 Q9UBN7 3/20 0.51
OPRL1 P41146 3/20 0.50
OPRM1 P35372 3/20 0.50
OPRD1 P41143 3/20 0.50
OPRK1 P41145 3/20 0.50
CYP2D6 P10635 1/20 0.47
CCR5 P51681 1/20 0.47
LMNA P02545 1/20 0.46
GAA P10253 1/20 0.46
ALOX15 P16050 1/20 0.46
TP53 P04637 1/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
MAPT P10636 1/20 0.45
GFER P55789 1/20 0.45
TDP1 Q9NUW8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18250748 0.84 CCR5 (0.58) OPRM1OPRD1OPRK1CYP2D6CCR5
SCHEMBL3448194 0.84 GAA (0.61) OPRM1OPRD1OPRK1CYP2D6CCR5
SCHEMBL7587030 0.82 CCR5 (0.54) JAK2JAK1OPRM1OPRD1OPRK1
SCHEMBL18250718 0.82 GAA (0.64) OPRM1OPRD1OPRK1CYP2D6CCR5
Hydrochloric Acid SCHEMBL4379304 0.81 CCR5 (0.53) JAK2JAK1OPRM1OPRD1OPRK1
SCHEMBL9673866 0.80 CCR5 (0.60) CYP2D6CCR5LMNAGAAALOX15
SCHEMBL14605232 0.79 JAK1 (0.69) JAK2JAK1GAAALOX15
SCHEMBL14605231 0.79 JAK1 (0.69) JAK2JAK1GAAALOX15
SCHEMBL13545208 0.77 CCR5 (0.51) OPRL1OPRM1OPRD1OPRK1CYP2D6
SCHEMBL739512 0.76 HDAC1 (0.49) HDAC1HDAC8HDAC6OPRL1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed