SCHEMBL3448194

SCHEMBL3448194

Cc1nc2ccccc2n1C1CCCC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.61
ALOX15 P16050 1/20 0.61
CYP2D6 P10635 2/20 0.61
CCR5 P51681 1/20 0.61
ALDH1A1 P00352 2/20 0.60
MAPT P10636 2/20 0.60
TP53 P04637 1/20 0.60
KDM4E B2RXH2 1/20 0.60
GFER P55789 1/20 0.60
TDP1 Q9NUW8 1/20 0.60
CCNT1 O60563 1/20 0.58
CDK9 P50750 1/20 0.58
LMNA P02545 2/20 0.56
L3MBTL1 Q9Y468 2/20 0.56
PRKACA P17612 3/20 0.55
RPS6KB1 P23443 3/20 0.55
GSK3B P49841 3/20 0.55
ROCK1 Q13464 3/20 0.55
OPRM1 P35372 2/20 0.53
OPRD1 P41143 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18250718 0.98 GAA (0.64) GAAALOX15CYP2D6CCR5ALDH1A1
SCHEMBL18250748 0.97 CCR5 (0.58) GAAALOX15CYP2D6CCR5ALDH1A1
SCHEMBL9673866 0.93 CCR5 (0.60) GAAALOX15CYP2D6CCR5ALDH1A1
SCHEMBL7587030 0.85 CCR5 (0.54) GAAALOX15CYP2D6CCR5ALDH1A1
SCHEMBL3732583 0.85 CCR5 (0.64) GAAALOX15CYP2D6CCR5LMNA
SCHEMBL10219470 0.85 CYP2D6 (0.54) GAAALOX15CYP2D6CCR5ALDH1A1
Hydrochloric Acid SCHEMBL4379304 0.84 CCR5 (0.53) GAAALOX15CYP2D6CCR5ALDH1A1
SCHEMBL763378 0.84 JAK2 (0.53) GAAALOX15CYP2D6CCR5ALDH1A1
SCHEMBL13545208 0.82 CCR5 (0.51) CYP2D6CCR5LMNAOPRM1OPRD1
Hydrochloric Acid SCHEMBL20958819 0.81 ALDH1A1 (0.48) GAAALOX15CYP2D6CCR5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9499529-B2 Therapeutic uses of curcumin analogs for treatment of prostate cancer CALIFORNIA STATE UNIVERSITY, FRESNO (US) 2016-11-22 US disclosed
US-7855211-B2 such as [5-(4-Ethyl-piperazin-1-ylmethyl)-pyridin-2-yl]-[5-fluoro-4-(7-fluoro-3-isopropyl-2-methyl-3H-benzoimidazol-5-yl)-pyrimidin-2-yl]-amine, useful in the treatment of cell proliferative diseases ELI LILLY AND COMPANY (US) 2010-12-21 US disclosed
US-20100160340-A1 such as [5-(4-Ethyl-piperazin-1-ylmethyl)-pyridin-2-yl]-[5-fluoro-4-(7-fluoro-3-isopropyl-2-methyl-3H-benzoimidazol-5-yl)-pyrimidin-2-yl]-amine, useful in the treatment of cell proliferative diseases ELI LILLY AND COMPANY 2010-06-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100160340-A1 such as [5-(4-Ethyl-piperazin-1-ylmethyl)-pyridin-2-yl]-[5-fluoro-4-(7-fluoro-3-isopropyl-2-methyl-3H-benzoimidazol-5-yl)-pyrimidin-2-yl]-amine, useful in the treatment of cell proliferative diseases MKI67, PKD1, CCNI GAA 1317/4885ALOX15 1568/4885CYP2D6 2996/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.