SCHEMBL763422

SCHEMBL763422

COCCCn1c([C@@H]2CCCN(C(=O)C[C@@H](Cc3ccc(-c4ccccc4)cc3)NC(=O)OC(C)(C)C)C2)nc2ccncc21

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 4/20 0.37
KCNH2 Q12809 3/20 0.37
CYP2D6 P10635 2/20 0.37
KLK5 Q9Y337 1/20 0.37
ACE P12821 1/20 0.36
NLRP3 Q96P20 2/20 0.36
HRH2 P25021 1/20 0.36
TP53 P04637 1/20 0.36
THRB P10828 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CHRM1 P11229 1/20 0.35
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
CYP3A4 P08684 5/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ATM Q13315 1/20 0.34
USP30 Q70CQ3 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL763858 0.93 KCNH2 (0.42) HRH1KCNH2CYP2D6KLK5ACE
SCHEMBL762527 0.92 NLRP3 (0.39) HRH1KCNH2CYP2D6KLK5NLRP3
SCHEMBL739362 0.92 HRH1 (0.40) HRH1KCNH2CYP2D6NLRP3TP53
SCHEMBL763874 0.90 HRH1 (0.39) HRH1KCNH2CYP2D6KLK5CHRM1
SCHEMBL739547 0.89 HRH1 (0.41) HRH1KCNH2CYP2D6KLK5HRH2
SCHEMBL739548 0.89 HRH1 (0.41) HRH1KCNH2CYP2D6KLK5HRH2
SCHEMBL16301222 0.89 HRH1 (0.38) HRH1KCNH2CYP2D6TP53THRB
SCHEMBL16301236 0.88 KCNH2 (0.47) HRH1KCNH2CYP2D6TP53SMN1; SMN2
SCHEMBL16301237 0.88 HRH1 (0.40) HRH1KCNH2CYP2D6KLK5CHRM1
SCHEMBL739119 0.88 HRH1 (0.39) HRH1KCNH2CYP2D6HRH2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed