SCHEMBL764081

SCHEMBL764081

CNC(C)c1ccc(F)c(F)c1F

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.39
CES1 P23141 2/20 0.39
HTR2A P28223 7/20 0.38
SLC6A4 P31645 7/20 0.38
KCNH2 Q12809 5/20 0.38
CYP2D6 P10635 1/20 0.35
NPC1 O15118 1/20 0.31
ADRA2A P08913 2/20 0.30
ADRA2B P18089 2/20 0.30
ADRA2C P18825 2/20 0.30
ADRA1A P35348 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL178631 0.81 HTR2A (0.40) HTR2ASLC6A4KCNH2CYP2D6
SCHEMBL26948996 0.81 CES2 (0.41) CES2CES1HTR2ASLC6A4KCNH2
SCHEMBL2668988 0.81 CES2 (0.41) CES2CES1HTR2ASLC6A4KCNH2
SCHEMBL17553266 0.77 CES2 (0.41) CES2CES1
SCHEMBL12049608 0.77 CES2 (0.44) CES2CES1NPC1ADRA1A
SCHEMBL178490 0.74 SLC6A4 (0.50) HTR2ASLC6A4KCNH2CYP2D6
SCHEMBL178501 0.74 SLC6A4 (0.39) HTR2ASLC6A4KCNH2CYP2D6
SCHEMBL9070739 0.74 SLC6A4 (0.50) HTR2ASLC6A4KCNH2CYP2D6
SCHEMBL24989671 0.73 CES2 (0.41) CES2CES1
SCHEMBL16956342 0.73 CES2 (0.41) CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8883824-B2 3-(4-aminophenyl)-2-furancarboxylic acid derivative and pharmaceutically acceptable salt thereof SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2014-11-11 US disclosed
EP-2431362-A1 3-(4-AMINOPHENYL)-2-FURANCARBOXYLIC ACID DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF Dainippon Sumitomo Pharma Co., Ltd. (JP) 2012-03-21 EP disclosed
WO-2010131669-A1 3-(4-AMINOPHENYL)-2-FURANCARBOXYLIC ACID DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF 大日本住友製薬株式会社 (JP) 2010-11-18 WO disclosed