SCHEMBL2668988

SCHEMBL2668988

CNC(C)c1cccc(F)c1F

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.41
CES1 P23141 2/20 0.41
HTR2A P28223 5/20 0.39
SLC6A4 P31645 5/20 0.39
CYP2D6 P10635 1/20 0.38
IDH1 O75874 4/20 0.37
ADRB1 P08588 1/20 0.36
ADRA2A P08913 1/20 0.36
ADRB3 P13945 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
KCNH2 Q12809 3/20 0.35
SOS1 Q07889 3/20 0.34
BCHE P06276 1/20 0.33
MAPKAPK2 P49137 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26948996 1.00 CES2 (0.41) CES2CES1HTR2ASLC6A4CYP2D6
SCHEMBL30634130 0.83 SLC6A4 (0.44) CES2CES1HTR2ASLC6A4CYP2D6
SCHEMBL2404369 0.83 SLC6A4 (0.44) CES2CES1HTR2ASLC6A4CYP2D6
SCHEMBL16254312 0.83 SLC6A4 (0.44) CES2CES1HTR2ASLC6A4CYP2D6
SCHEMBL23159244 0.82 CES2 (0.40) CES2CES1IDH1ADRB1ADRA2A
SCHEMBL26494862 0.82 SOS1 (0.43) HTR2ASLC6A4CYP2D6SOS1
SCHEMBL764081 0.81 CES2 (0.39) CES2CES1HTR2ASLC6A4CYP2D6
SCHEMBL22904344 0.80 HTR2A (0.42) HTR2ASLC6A4CYP2D6KCNH2SOS1
SCHEMBL25078726 0.80 HTR2A (0.42) HTR2ASLC6A4CYP2D6KCNH2SOS1
SCHEMBL26487709 0.80 CFD (0.45) HTR2ASLC6A4CYP2D6ADRB1ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022260441-A1 PREPARATION OF SUBSTITUTED 1,2-DIAMINOHETEROCYCLIC COMPOUND DERIVATIVES AND THEIR USE AS PHARMACEUTICAL AGENTS AVELOS THERAPEUTICS INC. (KR) 2022-12-15 WO disclosed
WO-2021055326-A1 AZOLE-FUSED PYRIDAZIN-3(2H)-ONE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2021-03-25 WO disclosed
US-8883824-B2 3-(4-aminophenyl)-2-furancarboxylic acid derivative and pharmaceutically acceptable salt thereof SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2014-11-11 US disclosed
EP-2431362-A1 3-(4-AMINOPHENYL)-2-FURANCARBOXYLIC ACID DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF Dainippon Sumitomo Pharma Co., Ltd. (JP) 2012-03-21 EP disclosed
WO-2010131669-A1 3-(4-AMINOPHENYL)-2-FURANCARBOXYLIC ACID DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF 大日本住友製薬株式会社 (JP) 2010-11-18 WO disclosed