SCHEMBL7642867

SCHEMBL7642867

CCc1cccc(N(CC)C(N)=Nc2ccc(C)cc2)c1

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 19/20 0.61
TP53 P04637 1/20 0.44
CYP2D6 P10635 1/20 0.44
TSHR P16473 1/20 0.44
THPO P40225 1/20 0.44
MTOR P42345 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7642451 0.88 SIGMAR1 (0.60) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL6720717 0.88 SIGMAR1 (0.62) SIGMAR1
SCHEMBL7615602 0.88 SIGMAR1 (0.54) SIGMAR1TP53
SCHEMBL6721400 0.88 SIGMAR1 (0.72) SIGMAR1
SCHEMBL6724260 0.86 SIGMAR1 (0.62) SIGMAR1
SCHEMBL6725057 0.77 SIGMAR1 (0.76) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL6719553 0.76 SIGMAR1 (1.00) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL6716625 0.75 SIGMAR1 (0.77) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL7647490 0.74 SIGMAR1 (0.78) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL6727463 0.74 SIGMAR1 (0.85) SIGMAR1TP53CYP2D6TSHRTHPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0517852-B1 TRI- AND TETRA-SUBSTITUTED GUANIDINES AND THEIR USE AS EXCITATORY AMINO ACID ANTAGONISTS OREGON STATE (US) 2002-07-10 EP claimed